SCHEMBL8329247

SCHEMBL8329247

C[Sn](C)(C)c1cncc(Cl)c1

nearest known ligand 0.39

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
HCAR2 Q8TDS4 1/20 0.39
CHRNB2 P17787 3/20 0.35
CHRNA4 P43681 3/20 0.35
HDAC8 Q9BY41 1/20 0.32
CHRNB4 P30926 1/20 0.32
CHRNA3 P32297 1/20 0.32
MKNK1 Q9BUB5 1/20 0.32
MKNK2 Q9HBH9 1/20 0.32
FGFR1 P11362 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL197638 0.73
SCHEMBL5952220 0.71 TSHR (0.50)
SCHEMBL12502235 0.70 CHRNB2 (0.33) HCAR2CHRNB2CHRNA4
SCHEMBL28044800 0.70
SCHEMBL30129770 0.70
Hydrochloric Acid SCHEMBL6069542 0.70
Water SCHEMBL28044737 0.70
Water SCHEMBL28044696 0.68 HCAR2 (0.48) HCAR2CHRNB2CHRNA4HDAC8CHRNB4
SCHEMBL31171067 0.67
SCHEMBL112244 0.67

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5922742-A NOVEL COMPOUNDS ACT AS ANTIINFLAMMATORY AGENTS, ANTIPYRETICS, AND ANALGESICS AND WOULD INHIBIT HORMONE-INDUCED UTERINE CONTRACTIONS WITHOUT MECHANISM-BASED SIDE EFFECTS MERCK FROSST CANADA (CA) 1999-07-13 US disclosed
EP-0900201-A1 PYRIDINYL-2-CYCLOPENTEN-1-ONES AS SELECTIVE CYCLOOXYGENASE-2 INHIBITORS MERCK FROSST CANADA INC. (CA) 1999-03-10 EP disclosed
WO-1997040012-A1 PYRIDINYL-2-CYCLOPENTEN-1-ONES AS SELECTIVE CYCLOOXYGENASE-2 INHIBITORS MERCK FROSST CANADA INC. (CA) 1997-10-30 WO disclosed