SCHEMBL8330131

SCHEMBL8330131

COc1cc2c(cc1OC)[C@H]1CN(C)CC[C@H]1N=C2c1ccc(NS(C)(=O)=O)cc1

nearest known ligand 0.78

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
PDE4D Q08499 2/20 0.78
PDE4A P27815 1/20 0.60
PDE4B Q07343 1/20 0.60
PDE4C Q08493 1/20 0.60
KDM1A O60341 5/20 0.40
ABCB1 P08183 1/20 0.39
CYP17A1 P05093 2/20 0.39
HTR7 P34969 2/20 0.37
HTR6 P50406 2/20 0.37
HTR1A P08908 1/20 0.37
HTR2A P28223 1/20 0.37
MAOA P21397 3/20 0.36
UTS2R Q9UKP6 2/20 0.36
MAOB P27338 1/20 0.36
MAPT P10636 2/20 0.36
ALDH1A1 P00352 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
IDO1 P14902 1/20 0.35
TDO2 P48775 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8326810 0.88 PDE4D (0.87) PDE4DPDE4APDE4BPDE4CMAPT
SCHEMBL8326816 0.88 PDE4D (0.87) PDE4DPDE4APDE4BPDE4CMAPT
Tolafentrine SCHEMBL159331 0.88 PDE4D (1.00) PDE4DPDE4APDE4BPDE4CHTR7
Tolafentrine SCHEMBL8326829 0.88 PDE4D (1.00) PDE4DPDE4APDE4BPDE4CHTR7
Tolafentrine SCHEMBL4450984 0.88 PDE4D (1.00) PDE4DPDE4APDE4BPDE4CHTR7
Tolafentrine SCHEMBL29992625 0.88 PDE4D (1.00) PDE4DPDE4APDE4BPDE4CHTR7
SCHEMBL7356412 0.87 PDE4D (0.86) PDE4DPDE4APDE4BPDE4CUTS2R
SCHEMBL7356403 0.87 PDE4D (0.86) PDE4DPDE4APDE4BPDE4CUTS2R
SCHEMBL7210383 0.86 PDE4D (0.69) PDE4DPDE4APDE4BPDE4CABCB1
SCHEMBL11843109 0.86 PDE4D (0.68) PDE4DPDE4APDE4BPDE4CUTS2R

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0528922-B1 NEW SULFONYL COMPOUNDS BYK GULDEN LOMBERG CHEM FAB (DE) 1999-06-16 EP claimed
US-5346904-A BRONCHODILATOR AGENTS BYK GULDEN LOMBERG CHEMISCHE FABRIK GMBH (DE) 1994-09-13 US claimed
EP-0528922-B1 NEW SULFONYL COMPOUNDS BYK GULDEN LOMBERG CHEM FAB (DE) 1999-06-16 EP disclosed
US-5346904-A BRONCHODILATOR AGENTS BYK GULDEN LOMBERG CHEMISCHE FABRIK GMBH (DE) 1994-09-13 US disclosed