SCHEMBL8330175

SCHEMBL8330175

Cc1cc(N)nc2c1CCCC2

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
NOS3 P29474 1/20 1.00
NOS1 P29475 1/20 1.00
NOS2 P35228 1/20 1.00
KDM4E B2RXH2 1/20 0.52
ACHE P22303 17/20 0.50
MEN1 O00255 1/20 0.48
MAPK1 P28482 1/20 0.48
KMT2A Q03164 1/20 0.48
BPTF Q12830 1/20 0.48
NPC1 O15118 1/20 0.47
RAB9A P51151 1/20 0.47
BCHE P06276 9/20 0.46
GRIN1 Q05586 9/20 0.46
GRIN2A Q12879 9/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30471705 0.96 NOS3 (0.92) NOS3NOS1NOS2KDM4EACHE
SCHEMBL527227 0.78 NOS3 (0.64) NOS3NOS1NOS2KDM4EACHE
SCHEMBL29621658 0.78 NOS3 (0.64) NOS3NOS1NOS2KDM4EACHE
SCHEMBL20417066 0.77 NOS3 (0.62) NOS3NOS1NOS2KDM4EACHE
SCHEMBL4926313 0.75 NOS3 (0.60) NOS3NOS1NOS2KDM4EACHE
SCHEMBL4928326 0.75 NOS3 (0.60) NOS3NOS1NOS2KDM4EACHE
SCHEMBL9753025 0.74 NOS3 (0.59) NOS3NOS1NOS2KDM4EACHE
SCHEMBL20416983 0.74 NOS3 (0.59) NOS3NOS1NOS2KDM4EACHE
SCHEMBL25807047 0.72 NOS3 (0.56) NOS3NOS1NOS2KDM4EACHE
SCHEMBL19998979 0.72 NOS3 (0.56) NOS3NOS1NOS2KDM4EACHE

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1290249-A Aminoguanidine hydrazone derivatives, process for producing the same and drugs thereof TAKEDA CHEMICAL INDUSTRIES LTD (JP) 2001-04-04 CN disclosed
US-5972975-A Substituted 2-aminopyridines as inhibitors of nitric oxide synthase MERCK & CO., INC. (US) 1999-10-26 US disclosed
WO-1996018616-A1 SUBSTITUTED 2-AMINOPYRIDINES AS INHIBITORS OF NITRIC OXIDE SYNTHASE MERCK & CO., INC. (US) 1996-06-20 WO disclosed
WO-1991017979-A1 PROCESS FOR THE PREPARATION OF 2-N-ACYLAMINOPYRIDINES AND 2-AMINOPYRIDINES FROM 5-OXOALKANENITRILE OXIMES DSM N.V. (NL) 1991-11-28 WO disclosed