SCHEMBL8330192

SCHEMBL8330192

O=CCC(NC(=O)c1ccccc1)(c1ccccc1)N1CCCCC1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTT P42858 2/20 0.44
GAA P10253 1/20 0.43
CYP2C9 P11712 2/20 0.40
MAPT P10636 4/20 0.39
ALDH1A1 P00352 4/20 0.39
SMN1; SMN2 Q16637 3/20 0.39
TSHR P16473 2/20 0.39
NPC1 O15118 2/20 0.39
RAB9A P51151 2/20 0.39
KMT2A Q03164 2/20 0.39
TP53 P04637 1/20 0.39
PKM P14618 1/20 0.39
NFKB1 P19838 1/20 0.39
NFKB2 Q00653 1/20 0.39
RELA Q04206 1/20 0.39
HPGD P15428 3/20 0.39
CYP2C19 P33261 2/20 0.39
CYP1A2 P05177 1/20 0.39
CTDSP1 Q9GZU7 1/20 0.38
LMNA P02545 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL703097 0.72 CYP2B6 (0.44) MAPTALDH1A1TSHRKMT2ANFKB1
SCHEMBL4508029 0.66 POLB (0.56) HTTGAACYP2C9MAPTALDH1A1
SCHEMBL27927957 0.64 CYP2B6 (0.44) MAPTTSHRKMT2ANFKB1LMNA
SCHEMBL17373911 0.64 POLB (0.58) HTTGAAALDH1A1KMT2AHPGD
SCHEMBL1072704 0.64 CYP2B6 (0.59) HTTGAAKMT2ALMNACYP2B6
SCHEMBL9134669 0.63 HDAC3 (0.52) GAACYP2C9MAPTALDH1A1SMN1; SMN2
SCHEMBL29190271 0.63 CYP3A4 (0.52) HTTGAACYP2C9MAPTALDH1A1
N-Piperidinobenzamide SCHEMBL696161 0.63 HTT (1.00) HTTGAACYP2C9MAPTALDH1A1
SCHEMBL9282775 0.63 HTT (1.00) HTTGAACYP2C9MAPTALDH1A1
SCHEMBL3174309 0.62 DRD4 (0.62) HTTGAACYP2C9ALDH1A1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5977101-A Benzimidazoles/Imidazoles Linked to a Fibrinogen Receptor Antagonist Template Having Vitronectin Receptor Antagonist Activity SMITHKLINE BEECHAM CORPORATION (US) 1999-11-02 US disclosed
EP-0869787-A4 VITRONECTIN RECEPTOR ANTAGONISTS SMITHKLINE BEECHAM CORP (US) 1999-03-24 EP disclosed
EP-0869787-A1 VITRONECTIN RECEPTOR ANTAGONISTS SMITHKLINE BEECHAM CORPORATION (US) 1998-10-14 EP disclosed
WO-1997024119-A1 VITRONECTIN RECEPTOR ANTAGONISTS SMITHKLINE BEECHAM CORPORATION (US) 1997-07-10 WO disclosed