SCHEMBL8330414

SCHEMBL8330414

C=C(OCC)[C@H](Cc1ccc2c(c1)NC(=O)[C@@H](CCC(=O)Nc1ncc[nH]1)O2)NC(=O)OC(C)(C)C

nearest known ligand 0.35

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
CCKAR P32238 1/20 0.34
CCKBR P32239 1/20 0.34
ITGB3 P05106 2/20 0.34
ITGAV P06756 2/20 0.34
HSD17B10 Q99714 3/20 0.33
TSHR P16473 2/20 0.33
THRB P10828 1/20 0.33
MEN1 O00255 2/20 0.33
KMT2A Q03164 2/20 0.33
USP2 O75604 1/20 0.33
GAA P10253 1/20 0.33
TP53 P04637 2/20 0.32
MAPT P10636 1/20 0.32
POLB P06746 1/20 0.32
SMN1; SMN2 Q16637 1/20 0.32
IDO1 P14902 1/20 0.32
ALOX15 P16050 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4850590 0.94 CCKAR (0.35) CCKARCCKBRITGB3ITGAVHSD17B10
SCHEMBL7163716 0.90 ACE (0.41) CCKARCCKBRITGB3ITGAVHSD17B10
SCHEMBL7163504 0.90 ACE (0.41) CCKARCCKBRITGB3ITGAVHSD17B10
SCHEMBL4681624 0.86 ITGB3 (0.36) ITGB3ITGAVHSD17B10TSHRTHRB
SCHEMBL4682248 0.86 ITGB3 (0.36) ITGB3ITGAVHSD17B10TSHRTHRB
SCHEMBL14143519 0.86 ITGB3 (0.36) ITGB3ITGAVHSD17B10TSHRTHRB
SCHEMBL14143487 0.86 TSHR (0.36) HSD17B10TSHRTHRBMEN1KMT2A
SCHEMBL14181804 0.84 TSHR (0.37) HSD17B10TSHRTHRBMEN1KMT2A
SCHEMBL4684103 0.84 ITGB3 (0.36) ITGB3ITGAVHSD17B10TSHRTHRB
SCHEMBL7163786 0.84 ITGB3 (0.36) CCKARCCKBRITGB3ITGAVHSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2004072054-A1 METHOD FOR THE PRODUCTION OF BICYCLIC AROMATIC AMINO ACIDS AND INTERMEDIATE PRODUCTS THEREOF MERCK PATENT GMBH (DE) 2004-08-26 WO disclosed