SCHEMBL8330978

SCHEMBL8330978

CC(C)Oc1ncc(N)cc1Br

nearest known ligand 0.35

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
CDK1 P06493 1/20 0.35
CCNB1 P14635 1/20 0.35
CCNA2 P20248 1/20 0.35
CDK2 P24941 1/20 0.35
CCNA1 P78396 1/20 0.35
ALOX5AP P20292 2/20 0.33
FEN1 P39748 2/20 0.33
MAPT P10636 2/20 0.32
NPSR1 Q6W5P4 1/20 0.32
GAA P10253 1/20 0.32
HTT P42858 1/20 0.31
KMT2A Q03164 1/20 0.31
MAP4K4 O95819 1/20 0.31
TLR8 Q9NR97 1/20 0.30
HRH4 Q9H3N8 1/20 0.30
SMN1; SMN2 Q16637 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3553372 0.79 LRRK2 (0.33) MAPT
SCHEMBL1558307 0.79 MAPT (0.41) ALOX5APFEN1MAPTNPSR1GAA
SCHEMBL31703952 0.78
SCHEMBL9379161 0.78 S1PR1 (0.37) CDK1CCNB1CCNA2CDK2CCNA1
SCHEMBL26693926 0.78 PLAU (0.39) MAP4K4SMN1; SMN2
SCHEMBL16248212 0.78 POLB (0.33)
SCHEMBL29837826 0.78 PLAU (0.39) MAP4K4SMN1; SMN2
SCHEMBL16046248 0.76 HPGD (0.38) CDK1CDK2MAPTGAAHTT
SCHEMBL789861 0.74 HTT (0.39) CDK1CCNB1CCNA2CDK2CCNA1
SCHEMBL7909807 0.74 PTGS2 (0.39) CDK1KMT2ASMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5929094-A NOVEL 3-((SUBSTITUTED) HETEROCYCLE),6-(SUBSTITUTED PHENYL)-1-OXASPIRO(4.4)NONANE DERIVATIVES; ANTAGONIZING THE EFFECT OF SUBSTANCE P BY ADMINISTERING TO BLOCK NEUROKININ-1 RECEPTORS; TREATING INFLAMMATION, MIGRAINE, EMESIS AND ASTHMA MERCK & CO., INC. (US) 1999-07-27 US disclosed
WO-1998017276-A1 HETEROARYL SPIROETHERCYCLOALKYL TACHYKININ RECEPTOR ANTAGONISTS MERCK & CO., INC. (US) 1998-04-30 WO disclosed