SCHEMBL8334973

SCHEMBL8334973

COC(=O)[C@H](Cc1ccc(O)cc1)NC(=O)c1ccccc1-c1ccccc1C(=O)N[C@@H](Cc1ccccc1)C(=O)N[C@@H](CC(C)C)C(=O)OC

nearest known ligand 0.60

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
TSHR P16473 1/20 0.60
IL1RN P18510 5/20 0.55
ERAP2 Q6P179 5/20 0.55
ERAP1 Q9NZ08 4/20 0.55
BIRC2 Q13490 1/20 0.53
ALDH1A1 P00352 1/20 0.52
THRB P10828 1/20 0.52
CYP2C9 P11712 1/20 0.52
CYP2C19 P33261 1/20 0.52
HSD17B10 Q99714 1/20 0.52
KDR P35968 1/20 0.51
NPY1R P25929 1/20 0.50
NPY4R P50391 1/20 0.50
CAPN1 P07384 1/20 0.50
ACE P12821 1/20 0.50
KCNA5 P22460 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8337125 0.94 TSHR (0.56) TSHRIL1RNERAP2ERAP1NPY1R
SCHEMBL8338416 0.85 TSHR (0.54) TSHRERAP2ERAP1ALDH1A1THRB
SCHEMBL8336881 0.85 TSHR (0.60) TSHRALDH1A1KDR
SCHEMBL8334773 0.85 TSHR (0.60) TSHRERAP2ERAP1ALDH1A1KDR
SCHEMBL4363977 0.83 TSHR (0.61) TSHRERAP2ERAP1ALDH1A1THRB
SCHEMBL4369419 0.83 TSHR (0.61) TSHRERAP2ERAP1ALDH1A1THRB
SCHEMBL13669588 0.82 TSHR (0.67) TSHRERAP2ERAP1ALDH1A1THRB
SCHEMBL11580063 0.82 TSHR (0.67) TSHRERAP2ERAP1ALDH1A1THRB
SCHEMBL4366475 0.82 TSHR (0.67) TSHRERAP2ERAP1ALDH1A1THRB
SCHEMBL13669590 0.82 TSHR (0.67) TSHRERAP2ERAP1ALDH1A1THRB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2004101494-A1 CALPAIN INHIBITORS CONSEJO SUPERIOR DE INVESTIGACIONES CIENTÍFICAS (ES) 2004-11-25 WO disclosed