SCHEMBL8334773

SCHEMBL8334773

COC(=O)[C@H](Cc1ccc(O)cc1)NC(=O)c1ccccc1-c1ccccc1C(=O)N[C@@H](Cc1ccc(O)cc1)C(=O)O

nearest known ligand 0.60

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 1/20 0.60
KDR P35968 1/20 0.58
LNPEP Q9UIQ6 2/20 0.57
MDM4 O15151 1/20 0.57
MDM2 Q00987 1/20 0.57
ELANE P08246 2/20 0.54
CDK2 P24941 2/20 0.53
ITGB1 P05556 3/20 0.52
ITGA4 P13612 3/20 0.52
ITGB7 P26010 3/20 0.52
CNR1 P21554 1/20 0.52
CNR2 P34972 1/20 0.52
TACR3 P29371 1/20 0.50
KDM4E B2RXH2 1/20 0.50
ALDH1A1 P00352 1/20 0.50
PKM P14618 1/20 0.50
ERAP2 Q6P179 1/20 0.49
ERAP1 Q9NZ08 1/20 0.49
KMT2A Q03164 1/20 0.49
NPSR1 Q6W5P4 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8279855 0.94 TSHR (0.53) TSHRKDRLNPEPMDM4MDM2
SCHEMBL8336881 0.93 TSHR (0.60) TSHRKDRLNPEPMDM4MDM2
SCHEMBL13940594 0.88 KDR (0.56) TSHRKDRLNPEPMDM4MDM2
SCHEMBL3988070 0.86 ALDH1A1 (0.55) ELANECNR1CNR2TACR3KDM4E
SCHEMBL8334980 0.85 ALDH1A1 (0.57) ELANECNR1CNR2TACR3KDM4E
SCHEMBL3975655 0.85 KDR (0.62) TSHRKDRLNPEPMDM4MDM2
SCHEMBL3975653 0.85 KDR (0.62) TSHRKDRLNPEPMDM4MDM2
SCHEMBL8334973 0.85 TSHR (0.60) TSHRKDRALDH1A1ERAP2ERAP1
SCHEMBL8337801 0.83 L3MBTL1 (0.60) ELANEITGB1ITGA4ITGB7KMT2A
SCHEMBL13940590 0.83 TSHR (0.56) TSHRKDRLNPEPMDM4MDM2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2004101494-A1 CALPAIN INHIBITORS CONSEJO SUPERIOR DE INVESTIGACIONES CIENTÍFICAS (ES) 2004-11-25 WO disclosed