SCHEMBL8335663

SCHEMBL8335663

O=C(Nc1ccccc1-c1ccccc1NC(=O)c1ccc2ccccc2c1)c1ccc2ccccc2c1

nearest known ligand 0.71

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 5/20 0.71
RAB9A P51151 5/20 0.71
DEGS1 O15121 2/20 0.64
GAA P10253 2/20 0.61
DHODH Q02127 2/20 0.58
KDM4E B2RXH2 1/20 0.58
TERT O14746 1/20 0.57
TOP1 P11387 1/20 0.57
MEN1 O00255 2/20 0.55
KMT2A Q03164 2/20 0.55
CASP3 P42574 1/20 0.55
SENP7 Q9BQF6 1/20 0.55
NR1H4 Q96RI1 2/20 0.54
SLC16A3 O15427 1/20 0.54
PPARG P37231 1/20 0.54
SIRT2 Q8IXJ6 1/20 0.54

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20541898 0.91 NPC1 (0.64) NPC1RAB9ADEGS1GAADHODH
SCHEMBL17915382 0.90 NPC1 (0.59) NPC1RAB9ADEGS1GAADHODH
SCHEMBL18347014 0.89 NPC1 (0.58) NPC1RAB9ADEGS1GAADHODH
SCHEMBL6627530 0.88 NPC1 (0.69) NPC1RAB9ADEGS1GAADHODH
SCHEMBL18347022 0.87 TRPV1 (0.61) NPC1RAB9ADEGS1GAADHODH
SCHEMBL18347006 0.86 NPC1 (0.56) NPC1RAB9ADEGS1GAADHODH
SCHEMBL18347008 0.86 SIRT2 (0.58) NPC1RAB9ADEGS1GAADHODH
SCHEMBL8337049 0.86 MEN1 (0.68) NPC1RAB9AMEN1KMT2ACASP3
SCHEMBL8335659 0.85 ALOX5 (0.65) NPC1RAB9ADEGS1MEN1KMT2A
SCHEMBL21870332 0.83 NPC1 (1.00) NPC1RAB9ADEGS1GAADHODH

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2004101494-A1 CALPAIN INHIBITORS CONSEJO SUPERIOR DE INVESTIGACIONES CIENTÍFICAS (ES) 2004-11-25 WO disclosed