SCHEMBL8337399

SCHEMBL8337399

Cc1cccc(COc2ccc(Br)cc2C(=O)N[C@@H](Cc2ccc(-c3ccccc3Oc3ccccc3)cc2)C(=O)C(C)O)c1

nearest known ligand 0.49

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
LRRK2 Q5S007 10/20 0.49
ABCG2 Q9UNQ0 1/20 0.44
KIFC1 Q9BW19 2/20 0.42
POLB P06746 2/20 0.39
CAPN1 P07384 1/20 0.39
MEN1 O00255 1/20 0.38
RECQL P46063 1/20 0.38
KMT2A Q03164 1/20 0.38
CTSB P07858 1/20 0.38
ITGB1 P05556 1/20 0.38
ITGA4 P13612 1/20 0.38
ITGB7 P26010 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8337386 0.94 LRRK2 (0.49) LRRK2ABCG2KIFC1POLBCAPN1
SCHEMBL5927497 0.93 LRRK2 (0.51) LRRK2ABCG2KIFC1POLBMEN1
SCHEMBL8337501 0.92 LRRK2 (0.47) LRRK2ABCG2KIFC1POLBCTSB
SCHEMBL5926743 0.91 ABCG2 (0.52) LRRK2ABCG2KIFC1POLBMEN1
SCHEMBL8337545 0.86 LRRK2 (0.38) LRRK2ABCG2KIFC1POLBITGB1
SCHEMBL5927425 0.85 KIFC1 (0.50) LRRK2ABCG2KIFC1POLBMEN1
SCHEMBL8337242 0.85 LRRK2 (0.37) LRRK2ABCG2KIFC1POLBCAPN1
SCHEMBL5927055 0.85 KIFC1 (0.55) LRRK2ABCG2KIFC1MEN1RECQL
SCHEMBL8337866 0.85 PTPN11 (0.44) LRRK2ABCG2POLBITGB1ITGA4
SCHEMBL5926387 0.84 ABCG2 (0.56) LRRK2ABCG2KIFC1POLBMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2004014844-A2 ARYL AND HETEROARYL COMPOUNDS AND METHODS TO MODULATE COAGULATION TRANSTECH PHARMA, INC. (US) 2004-02-19 WO disclosed