SCHEMBL8338729

SCHEMBL8338729

CC(O)C(=O)[C@H](Cc1ccc(-c2ccccc2)cc1)NC(=O)c1cc(Br)ccc1OCc1ccc(OCc2ccccc2)c(OCc2ccccc2)c1

nearest known ligand 0.49

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
KIFC1 Q9BW19 2/20 0.49
ABCG2 Q9UNQ0 1/20 0.49
LRRK2 Q5S007 10/20 0.48
SMPD1 P17405 1/20 0.45
CTSB P07858 2/20 0.44
POLB P06746 2/20 0.44
LMNA P02545 1/20 0.44
KDM4E B2RXH2 1/20 0.43
ALDH1A1 P00352 1/20 0.43
HPGD P15428 1/20 0.43
CTSS P25774 1/20 0.41
CAPN1 P07384 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8338624 0.93 LRRK2 (0.49) KIFC1ABCG2LRRK2
SCHEMBL4829673 0.90 KIFC1 (0.60) KIFC1ABCG2LRRK2POLBLMNA
SCHEMBL4829669 0.90 KIFC1 (0.60) KIFC1ABCG2LRRK2POLBLMNA
SCHEMBL4827862 0.89 ABCG2 (0.59) KIFC1ABCG2LRRK2SMPD1
SCHEMBL4827858 0.89 ABCG2 (0.59) KIFC1ABCG2LRRK2SMPD1
SCHEMBL8337501 0.87 LRRK2 (0.47) KIFC1ABCG2LRRK2SMPD1CTSB
SCHEMBL8337386 0.87 LRRK2 (0.49) KIFC1ABCG2LRRK2POLBLMNA
SCHEMBL4831380 0.86 KIFC1 (0.64) KIFC1ABCG2LRRK2POLBLMNA
SCHEMBL4831384 0.86 KIFC1 (0.64) KIFC1ABCG2LRRK2POLBLMNA
SCHEMBL4827793 0.85 ABCG2 (0.62) KIFC1ABCG2LRRK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2004014844-A2 ARYL AND HETEROARYL COMPOUNDS AND METHODS TO MODULATE COAGULATION TRANSTECH PHARMA, INC. (US) 2004-02-19 WO disclosed