SCHEMBL8339745

SCHEMBL8339745

Cc1ccc(OCC(=O)OCCN(C)C)cc1-c1nsc2ccc(-n3c(=O)cc(C(F)(F)F)n(C)c3=O)cc12

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 1/20 0.35
CYP3A4 P08684 1/20 0.35
CYP2C19 P33261 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
BLM P54132 1/20 0.35
PMP22 Q01453 1/20 0.35
HPGD P15428 1/20 0.34
TP53 P04637 2/20 0.31
MEN1 O00255 1/20 0.30
KMT2A Q03164 1/20 0.30
GAK O14976 1/20 0.30
EGFR P00533 1/20 0.30
ERBB2 P04626 1/20 0.30
JAK1 P23458 1/20 0.30
TTK P33981 1/20 0.30
TXK P42681 1/20 0.30
BLK P51451 1/20 0.30
JAK3 P52333 1/20 0.30
BTK Q06187 1/20 0.30
ITK Q08881 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7467248 0.90 TP53 (0.32) HPGDTP53
SCHEMBL7459571 0.87 AGER (0.35) HPGDMEN1KMT2A
SCHEMBL8339743 0.87 ESR1 (0.30) CYP1A2CYP3A4CYP2C19SMN1; SMN2
SCHEMBL7461743 0.85
SCHEMBL7460145 0.83 MEN1 (0.33) MEN1KMT2AMGLL
SCHEMBL8100008 0.82 MAPT (0.34)
SCHEMBL7454798 0.81 PPARD (0.35) HPGDMEN1KMT2A
SCHEMBL7459631 0.80 AR (0.36) SMN1; SMN2
SCHEMBL7458117 0.80 POLB (0.36) SMN1; SMN2HPGDMEN1KMT2A
SCHEMBL7463607 0.80 KMT2A (0.37) CYP3A4CYP2C19SMN1; SMN2TP53MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1999014216-A1 SUBSTITUTED 3(-1,2-BENZISOTHIAZOL OR ISOXAZOL-5 YL)-SUBSTITUTED PYRIMIDINE AS HERBICIDES AMERICAN CYANAMID COMPANY (US) 1999-03-25 WO disclosed