SCHEMBL8340318

SCHEMBL8340318

CNCc1cccc(Cl)n1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 2/20 0.42
TP53 P04637 1/20 0.42
NPSR1 Q6W5P4 1/20 0.41
PDCD1 Q15116 2/20 0.40
CD274 Q9NZQ7 2/20 0.40
MBOAT4 Q96T53 1/20 0.39
CXCR4 P61073 1/20 0.38
CYP3A4 P08684 2/20 0.38
TSHR P16473 1/20 0.38
ALDH1A1 P00352 3/20 0.37
MAPT P10636 2/20 0.35
GAA P10253 2/20 0.35
HPGD P15428 1/20 0.35
AGTR1 P30556 1/20 0.35
IDH1 O75874 1/20 0.35
IDH2 P48735 1/20 0.35
HTR3E A5X5Y0 1/20 0.34
HTR3B O95264 1/20 0.34
HTR3A P46098 1/20 0.34
HTR3D Q70Z44 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL523614 0.84 NPSR1 (0.54) KDM4ETP53NPSR1CXCR4CYP3A4
SCHEMBL24142565 0.83 CYP3A4 (0.40) NPSR1CD274MBOAT4CXCR4CYP3A4
SCHEMBL5046126 0.80 HRH3 (0.52) MBOAT4ALDH1A1MAPTGAAHPGD
SCHEMBL24254425 0.79 CYP3A4 (0.38) KDM4ENPSR1MBOAT4CXCR4CYP3A4
SCHEMBL29791992 0.77 SMN1; SMN2 (0.53) NPSR1MBOAT4CXCR4CYP3A4SMN1; SMN2
SCHEMBL2476858 0.77 SMN1; SMN2 (0.53) NPSR1MBOAT4CXCR4CYP3A4SMN1; SMN2
SCHEMBL7333040 0.77 CXCR4 (0.52) KDM4ETP53NPSR1CXCR4CYP3A4
SCHEMBL17813438 0.76 MALT1 (0.42) KDM4ENPSR1PDCD1CD274CYP3A4
SCHEMBL17117536 0.76 NPSR1 (0.77) KDM4ENPSR1CYP3A4ALDH1A1MAPT
SCHEMBL943445 0.76

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109320505-B Preparation and application of halogenated butenolide compound with insecticidal activity 海利尔药业集团股份有限公司 2022-08-02 CN disclosed
EP-2661428-B1 QUINOXALINES AND AZA-QUINOXALINES AS CRTH2 RECEPTOR MODULATORS MERCK SHARP & DOHME (US) 2017-06-07 EP disclosed
WO-2004024728-A2 PYRAZOLO[3,4-B]PYRIDINE COMPOUNDS, AND THEIR USE AS PHOSPHODIESTERASE INHIBITORS GLAXO GROUP LIMITED (GB) 2004-03-25 WO disclosed