SCHEMBL8340329

SCHEMBL8340329

Cc1cc(C)cc(C(=O)c2c(C(C)C)c(=O)[nH]c(=O)n2CCC2CC=CC2)c1

nearest known ligand 0.47

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 3/20 0.36
MEN1 O00255 2/20 0.36
TDP1 Q9NUW8 1/20 0.36
TP53 P04637 1/20 0.32
MAPT P10636 1/20 0.32
GRIN1 Q05586 1/20 0.31
GRIN2B Q13224 1/20 0.31
ALDH1A1 P00352 1/20 0.30
SMN1; SMN2 Q16637 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7071878 0.91 KMT2A (0.38) KMT2AMEN1TDP1GRIN1GRIN2B
SCHEMBL675171 0.89 KMT2A (0.35) KMT2AMEN1TDP1GRIN1GRIN2B
SCHEMBL7070169 0.86 KMT2A (0.36) KMT2AMEN1TDP1TP53MAPT
SCHEMBL12752183 0.85 KMT2A (0.47) KMT2AMEN1TDP1TP53MAPT
SCHEMBL2468222 0.85 TDP1 (0.33) KMT2AMEN1TDP1GRIN1GRIN2B
SCHEMBL12752190 0.84 KMT2A (0.39) KMT2AMEN1TDP1TP53MAPT
SCHEMBL674037 0.84 GRIN1 (0.42) KMT2AMEN1TDP1GRIN1GRIN2B
SCHEMBL12752179 0.83 KMT2A (0.41) KMT2AMEN1TDP1TP53MAPT
SCHEMBL8340328 0.83 TP53 (0.33) KMT2AMEN1TDP1TP53MAPT
SCHEMBL12752193 0.82 KMT2A (0.38) KMT2AMEN1TDP1TP53MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5922727-A 1-((SUBSTITUTED)CYCLOALK(EN)YLALKYL)-6-((SUB)PHENYL(CARBONYL, SULFIDE, OR OXO))-2,4-PYRIMIDINEDIONE DERIVATIVES HAVING SUPERIOR ANTIVIRAL ACTIVITIES; HIV SAMJIN PHARMACEUTICAL CO., LTD (KR) 1999-07-13 US disclosed