SCHEMBL8344819

SCHEMBL8344819

CCOC(=O)C[C@@]1(CN)C[C@H]2CC[C@H]2C1

nearest known ligand 0.38

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 1/20 0.38
GAA P10253 2/20 0.36
MGAM O43451 1/20 0.36
SI P14410 1/20 0.36
MGAM2 Q2M2H8 1/20 0.36
KMT2A Q03164 2/20 0.36
L3MBTL1 Q9Y468 1/20 0.36
EPHX2 P34913 2/20 0.35
ALDH1A1 P00352 3/20 0.34
TRPA1 O75762 1/20 0.34
SMYD3 Q9H7B4 1/20 0.33
ALOX15 P16050 1/20 0.32
CTDSP1 Q9GZU7 1/20 0.32
LMNA P02545 1/20 0.31
CHRM1 P11229 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14559622 1.00 CYP1A2 (0.38) CYP1A2GAAMGAMSIMGAM2
SCHEMBL8333639 0.85 CYP1A2 (0.39) CYP1A2GAAMGAMSIMGAM2
SCHEMBL14559647 0.83 CYP1A2 (0.40) CYP1A2GAAMGAMSIMGAM2
Pd-217014 SCHEMBL29539699 0.83 TSHR (0.35) CYP1A2GAAMGAMSIMGAM2
Pd-217014 SCHEMBL8306389 0.83 TSHR (0.35) CYP1A2GAAMGAMSIMGAM2
SCHEMBL18573883 0.80 CYP1A2 (0.44) CYP1A2GAAMGAMSIMGAM2
SCHEMBL14559623 0.80 KMT2A (0.33) GAAMGAMSIMGAM2KMT2A
SCHEMBL8345214 0.80 KMT2A (0.33) GAAMGAMSIMGAM2KMT2A
SCHEMBL16349096 0.78 EPHX2 (0.35) CYP1A2GAAMGAMSIMGAM2
SCHEMBL23960624 0.78 CYP1A2 (0.36) CYP1A2GAAMGAMSIMGAM2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1506955-B1 Bicyclic amino acids as pharmaceuticals agents WARNER LAMBERT CO (US) 2007-03-28 EP disclosed
US-7189747-B2 Method of treating noninflammatory cartilage damage WARNER-LAMBERT COMPANY (US) 2007-03-13 US disclosed
US-7189747-B2 Method of treating noninflammatory cartilage damage WARNER-LAMBERT COMPANY (US) 2007-03-13 US disclosed
WO-2003063845-A1 ALPHA 2 DELTA LIGANDS TO TREAT TINNITUS WARNER-LAMBERT COMPANY LLC (US) 2003-08-07 WO disclosed