SCHEMBL8344972

SCHEMBL8344972

CC(C)Cn1c(N)nc2c(=O)[nH]c(N)nc21

nearest known ligand 0.60

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
PNP P00491 9/20 0.60
HPRT1 P00492 5/20 0.43
KDM4E B2RXH2 1/20 0.41
NPSR1 Q6W5P4 1/20 0.41
DHFR P00374 1/20 0.40
PDE5A O76074 1/20 0.39
PDE4A P27815 1/20 0.39
PDE4B Q07343 1/20 0.39
PDE4C Q08493 1/20 0.39
PDE4D Q08499 1/20 0.39
XDH P47989 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL8341140 0.98 PNP (0.59) PNPHPRT1KDM4ENPSR1DHFR
SCHEMBL8344233 0.85 PNP (0.65) PNPHPRT1DHFR
Hydrochloric Acid SCHEMBL8345210 0.84 PNP (0.64) PNPHPRT1DHFR
SCHEMBL8587243 0.77 PNP (0.44) PNPHPRT1KDM4ENPSR1DHFR
SCHEMBL8344073 0.77 PNP (0.65) PNPHPRT1
SCHEMBL10871645 0.75 PNP (0.60) PNPHPRT1
Hydrochloric Acid SCHEMBL8341747 0.75 PNP (0.64) PNPHPRT1
SCHEMBL12820649 0.74 PNP (0.57) PNPDHFRXDH
SCHEMBL10872975 0.74 PNP (0.73) PNPHPRT1
SCHEMBL5503495 0.74 PNP (0.60) PNPHPRT1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5912252-A Purine and guanine derivatives as PNP inhibitors DARWIN DISCOVERY LIMITED (GB) 1999-06-15 US claimed
US-5912252-A Purine and guanine derivatives as PNP inhibitors DARWIN DISCOVERY LIMITED (GB) 1999-06-15 US disclosed