SCHEMBL8347367

SCHEMBL8347367

COc1ccc(C2CCC(c3ccc(OC)cc3)C2CO)cc1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM1A O60341 4/20 0.52
MAOA P21397 2/20 0.52
MAOB P27338 2/20 0.52
HTR2C P28335 1/20 0.49
MEN1 O00255 1/20 0.45
KMT2A Q03164 1/20 0.45
SLC6A2 P23975 2/20 0.41
SLC6A4 P31645 2/20 0.41
SLC6A3 Q01959 2/20 0.41
DRD2 P14416 1/20 0.41
RAB9A P51151 1/20 0.41
CA12 O43570 1/20 0.41
CA1 P00915 1/20 0.41
CA2 P00918 1/20 0.41
CA7 P43166 1/20 0.41
CA9 Q16790 1/20 0.41
CA14 Q9ULX7 1/20 0.41
TUBB4A P04350 1/20 0.41
TUBB P07437 1/20 0.41
TUBA3C P0DPH7 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16585495 0.78 HTR2C (0.67) KDM1AMAOAMAOBHTR2CDRD2
SCHEMBL16585494 0.78 HTR2C (0.67) KDM1AMAOAMAOBHTR2CDRD2
SCHEMBL19262122 0.78 HTR2C (0.67) KDM1AMAOAMAOBHTR2CDRD2
SCHEMBL17985307 0.78 HTR2C (0.67) KDM1AMAOAMAOBHTR2CDRD2
SCHEMBL8939863 0.77 HTR2C (0.49) KDM1AMAOAMAOBHTR2CMEN1
SCHEMBL16591168 0.76 KDM1A (0.64) KDM1AMAOAMAOBHTR2CMEN1
SCHEMBL18587035 0.76 KMT2A (0.45) MEN1KMT2ASLC6A2SLC6A4SLC6A3
SCHEMBL18587037 0.76 KMT2A (0.45) MEN1KMT2ASLC6A2SLC6A4SLC6A3
SCHEMBL27097274 0.76 HTR2C (0.47) KDM1AMAOAMAOBHTR2CMEN1
SCHEMBL16747456 0.75 KDM1A (0.47) KDM1AMAOAMAOBHTR2CTDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0693051-B1 CYCLOPENTENE AND CYCLOPENTANE DERIVATIVES AS ENDOTHELIN RECEPTOR ANTAGONISTS SMITHKLINE BEECHAM CORP (US) 1999-11-03 EP disclosed
US-5929116-A VASODILATOR; HYPOTENSIVE AGENT SMITHKLINE BEECHAM CORPORATION (US) 1999-07-27 US disclosed
WO-1994024084-A1 CYCLOPENTENE DERIVATIVES AS ENDOTHELIN RECEPTOR ANTAGONISTS SMITHKLINE BEECHAM CORPORATION (US) 1994-10-27 WO disclosed