SCHEMBL8347635

SCHEMBL8347635

CCCc1c(N2CCC(c3noc4cc(F)ccc34)CC2)ccc2c1C(=O)NC2=O

nearest known ligand 0.54

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
DRD2 P14416 8/20 0.54
SLC6A4 P31645 1/20 0.54
HTR2C P28335 11/20 0.49
HTR2A P28223 8/20 0.49
HTR1A P08908 1/20 0.49
DRD1 P21728 1/20 0.49
DRD3 P35462 1/20 0.49
HTR6 P50406 1/20 0.49
ACHE P22303 2/20 0.48
SCD O00767 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL8348525 0.99 DRD2 (0.53) DRD2SLC6A4HTR2CHTR2AHTR1A
SCHEMBL8345318 0.95 DRD2 (0.52) DRD2SLC6A4HTR2CHTR2AHTR1A
Hydrochloric Acid SCHEMBL8350488 0.94 DRD2 (0.52) DRD2SLC6A4HTR2CHTR2AHTR1A
SCHEMBL8345682 0.93 HTR2C (0.57) DRD2SLC6A4HTR2CHTR2AHTR1A
Hydrochloric Acid SCHEMBL8463604 0.92 HTR2C (0.56) DRD2SLC6A4HTR2CHTR2AHTR1A
Fumaric Acid SCHEMBL8350179 0.87 HTR2C (0.51) DRD2SLC6A4HTR2CHTR2AHTR1A
Fumaric Acid SCHEMBL8350178 0.87 HTR2C (0.51) DRD2SLC6A4HTR2CHTR2AHTR1A
SCHEMBL8648906 0.86 DRD2 (0.51) DRD2SLC6A4HTR2CHTR2AHTR1A
SCHEMBL8345401 0.85 HTR2C (0.54) DRD2SLC6A4HTR2CHTR2AHTR1A
Hydrochloric Acid SCHEMBL8566104 0.85 HTR2C (0.54) DRD2SLC6A4HTR2CHTR2AHTR1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 12 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5919798-A USEFUL AS ANTIPSYCHOTIC AND ANALGESIC AGENTS. HOECHST MARION ROUSSEL, INC. (US) 1999-07-06 US disclosed
US-5889035-A 1-(Arylthioalkyl, arylaminoalkyl or arylmethylenealkyl)-3-(heteroaryl) pyrrolidines and related compounds useful as antipsychotics and analgesics HOECHST MARION ROUSSEL, INC. (US) 1999-03-30 US disclosed
US-5889004-A PSYCHOLOGICAL DISORDERS, ANALGESICS HOECHST MARION ROUSSEL, INC. (US) 1999-03-30 US disclosed
US-5874435-A PSYCHOLOGICAL DISORDERS; ANALGESICS HOECHST MARION ROUSSEL, INC. (US) 1999-02-23 US disclosed
US-5854243-A 3-heteroaryl-1-pyrrolidinealkylthiols and derivatives thereof and their therapeutic utility HOECHST-ROUSSEL PHARMACEUTICALS, INC. (US) 1998-12-29 US disclosed
US-5854263-A 1- (1,4-benzodioxanyl)alkyl!-3-(heteroaryl) pyrrolidines and related compounds and their therapeutic utility HOECHST MARION ROUSSEL, INC. (US) 1998-12-29 US disclosed
US-5843977-A (3-heteroaryl-1-pyrrolidinyl) alkoxy!-3,4-dihydro-1(2H)-naphthalenones and related compounds and their therapeutic utility HOECHST MARION ROSUEEL, INC. 1998-12-01 US disclosed
US-5843949-A 1-(1H-indolyloxyalkyl)-4-(heteroaryl)piperazines and related compounds useful as antipsychotics and analgesics HOECHST MARION ROUSSEL, INC. 1998-12-01 US disclosed
US-5840727-A ANTIPSYCHOTICS, ANALGESICS AVENTIS PHARMACEUTICALS INC. 1998-11-24 US disclosed
US-5811430-A 1 (2-pyrimidinyloxy) alkyl!-4- (heteroaryl) Piperidines and related compounds and their therapeutic utility HOECHST MARION ROUSSEL, INC. 1998-09-22 US disclosed
US-5811435-A 2- (4-heteroaryl-1-piperidinyl)alkyl!-1,3-dioxanes and related compounds and their therapeutic utility HOECHST MARION RUSSEL, INC. 1998-09-22 US disclosed
US-5776963-A ANTIPSYCHOTIC AGENTS HOECHST MARION ROUSSEL, INC. (US) 1998-07-07 US disclosed