SCHEMBL8347752

SCHEMBL8347752

CCn1c(=O)c2ccccc2n(CCN(C)C)c1=O

nearest known ligand 0.57

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
MAPK8 P45983 1/20 0.55
TOP2A P11388 1/20 0.54
HDAC1 Q13547 1/20 0.53
ALDH1A1 P00352 3/20 0.52
KDM4E B2RXH2 2/20 0.52
PGR P06401 3/20 0.51
KMT2A Q03164 2/20 0.51
MPO P05164 1/20 0.50
HAVCR2 Q8TDQ0 1/20 0.50
HTR6 P50406 1/20 0.50
NPY5R Q15761 2/20 0.47
CNR2 P34972 1/20 0.47
RORA P35398 1/20 0.47
RORC P51449 1/20 0.47
RORB Q92753 1/20 0.47
SMN1; SMN2 Q16637 1/20 0.46
TDP1 Q9NUW8 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12963546 0.91 PGR (0.59) TOP2AHDAC1ALDH1A1KDM4EPGR
SCHEMBL6295469 0.85 MAPK8 (0.57) MAPK8ALDH1A1KDM4EPGRKMT2A
SCHEMBL12933336 0.85 TOP2A (0.51) TOP2AHDAC1ALDH1A1KDM4EPGR
SCHEMBL6362477 0.84 PGR (0.68) MAPK8HDAC1ALDH1A1KDM4EPGR
SCHEMBL30485670 0.84 PGR (0.68) MAPK8HDAC1ALDH1A1KDM4EPGR
SCHEMBL25936308 0.83 TOP2A (0.58) TOP2AHDAC1ALDH1A1KDM4EPGR
SCHEMBL6295236 0.82 MAPK8 (0.55) MAPK8ALDH1A1KDM4EPGRKMT2A
SCHEMBL12963428 0.81 PGR (0.61) MAPK8ALDH1A1KDM4EPGRKMT2A
SCHEMBL22201345 0.80 PGR (0.72) MAPK8TOP2AHDAC1PGRKMT2A
SCHEMBL17241700 0.79 HDAC1 (0.60) HDAC1ALDH1A1KMT2AHTR6TDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2004069823-A1 INHIBITORS OF HISTONE DEACETYLASE METHYLGENE, INC. (CA) 2004-08-19 WO disclosed
WO-2003024448-A2 INHIBITORS OF HISTONE DEACETYLASE METHYLGENE, INC. (CA) 2003-03-27 WO disclosed