SCHEMBL8348489

SCHEMBL8348489

Cc1cccc(CN=C=S)c1Cl

nearest known ligand 0.42

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
GABRA1 P14867 2/20 0.42
GABRB2 P47870 2/20 0.42
MIF P14174 10/20 0.41
TRPA1 O75762 3/20 0.41
ALDH1A1 P00352 2/20 0.41
CYP3A4 P08684 1/20 0.41
HPGD P15428 1/20 0.41
KEAP1 Q14145 2/20 0.38
NFE2L2 Q16236 2/20 0.38
CYP2E1 P05181 1/20 0.32
CYP2A6 P11509 1/20 0.32
HIF1A Q16665 1/20 0.32
CYP2A13 Q16696 1/20 0.32
EPAS1 Q99814 1/20 0.32
SLC6A4 P31645 2/20 0.32
CYP2D6 P10635 1/20 0.32
SLC6A2 P23975 1/20 0.32
SLC6A3 Q01959 1/20 0.32
PNMT P11086 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2564569 0.81 MIF (0.52) GABRA1GABRB2MIFTRPA1ALDH1A1
SCHEMBL8762257 0.80 MIF (0.42) GABRA1GABRB2MIFTRPA1ALDH1A1
SCHEMBL12458267 0.79 MIF (0.41) GABRA1GABRB2MIFTRPA1ALDH1A1
SCHEMBL14926027 0.76 MIF (0.45) GABRA1GABRB2MIFTRPA1ALDH1A1
SCHEMBL2141390 0.74 MIF (0.62) GABRA1GABRB2MIFTRPA1ALDH1A1
SCHEMBL29616337 0.74 MIF (0.62) GABRA1GABRB2MIFTRPA1ALDH1A1
SCHEMBL1457250 0.73 MIF (0.52) GABRA1GABRB2MIFTRPA1ALDH1A1
SCHEMBL14692301 0.72 KEAP1 (0.37) GABRA1GABRB2MIFTRPA1ALDH1A1
SCHEMBL2947684 0.71 MIF (0.46) GABRA1GABRB2MIFTRPA1ALDH1A1
SCHEMBL14024290 0.71 KAT2B (0.35) SLC6A4CYP2D6SLC6A2SLC6A3PNMT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7345065-B2 Methods and compositions for alleviating pain ALLERGAN, INC. (US) 2008-03-18 US disclosed
US-7345065-B2 Methods and compositions for alleviating pain ALLERGAN, INC. (US) 2008-03-18 US disclosed
WO-2003099289-A2 COMPOSITIONS AND THEIR USES FOR ALLEVIATING PAIN ALLERGAN, INC. (US) 2003-12-04 WO disclosed