SCHEMBL8348672

SCHEMBL8348672

NS(=O)(=O)c1ccccc1-c1c(-c2ccccc2)noc1CO

nearest known ligand 0.67

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 9/20 0.67
F2 P00734 3/20 0.48
F10 P00742 3/20 0.48
PTGS1 P23219 3/20 0.45
CA12 O43570 3/20 0.45
CA1 P00915 3/20 0.45
CA2 P00918 3/20 0.45
CA9 Q16790 3/20 0.45
MT-CO2 P00403 2/20 0.45
LMNA P02545 1/20 0.45
CA3 P07451 1/20 0.45
ADRB2 P07550 1/20 0.45
ADRB1 P08588 1/20 0.45
CYP3A4 P08684 1/20 0.45
ADORA3 P0DMS8 1/20 0.45
CHRM1 P11229 1/20 0.45
ADRA2B P18089 1/20 0.45
CA4 P22748 1/20 0.45
CA6 P23280 1/20 0.45
SLC6A2 P23975 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8476340 0.90 PTGS2 (0.55) PTGS2F2F10PTGS1CA12
SCHEMBL8477420 0.88 PTGS2 (0.56) PTGS2F2F10PTGS1CA12
SCHEMBL8475898 0.87 PTGS2 (0.61) PTGS2F2F10PTGS1CA12
SCHEMBL8473427 0.87 PTGS2 (0.51) PTGS2F2F10PTGS1CA12
SCHEMBL8476348 0.85 PTGS2 (0.49) PTGS2F2F10PTGS1CA12
SCHEMBL8474220 0.85 PTGS2 (0.53) PTGS2F2F10PTGS1CA12
SCHEMBL8479943 0.85 PTGS2 (0.49) PTGS2F2F10PTGS1CA12
SCHEMBL8473752 0.85 PTGS2 (0.50) PTGS2F2F10PTGS1CA12
SCHEMBL7963617 0.84 PTGS2 (0.49) PTGS2F2F10PTGS1CA12
SCHEMBL8480486 0.84 PTGS2 (0.48) PTGS2F2F10PTGS1CA12

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5932598-A NOVEL SUBSTITUTED SULFONAMIDE COMPOUNDS USEFUL AS PRODRUGS; ADMINISTERING TO TREAT INFLAMMATION-ASSOCIATED PAIN DUE TO CANCER, DENTAL PAIN; CYCLOOXYGENASE-2 INHIBITORS G. D. SEARLE & CO. (US) 1999-08-03 US disclosed
US-5859257-A ANTIINFLAMMATORY, ANTIARTHRITIC AGENTS G. D. SEARLE & CO. (US) 1999-01-12 US disclosed