SCHEMBL8353071

SCHEMBL8353071

Cn1c(=O)c2c(nc(N3CCCC3)n2Cc2ccccc2Br)n(C)c1=O

nearest known ligand 0.74

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 7/20 0.74
NPSR1 Q6W5P4 4/20 0.74
TSHR P16473 3/20 0.74
LMNA P02545 2/20 0.74
HTT P42858 2/20 0.74
MEN1 O00255 1/20 0.74
USP2 O75604 1/20 0.74
MAPT P10636 1/20 0.74
KMT2A Q03164 1/20 0.74
MAOB P27338 3/20 0.70
ADORA2A P29274 3/20 0.70
DPP4 P27487 4/20 0.63
L3MBTL1 Q9Y468 2/20 0.63
PCSK9 Q8NBP7 1/20 0.60
SMN1; SMN2 Q16637 2/20 0.59
CYP3A4 P08684 1/20 0.59
CYP2C9 P11712 1/20 0.59
CYP2C19 P33261 1/20 0.59
MAPK1 P28482 1/20 0.59
RECQL P46063 1/20 0.59

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5639692 0.91 DPP4 (0.72) ALDH1A1NPSR1TSHRLMNAHTT
SCHEMBL4667706 0.88 DPP4 (0.73) ALDH1A1NPSR1TSHRLMNAHTT
SCHEMBL555311 0.87 DPP4 (0.78) ALDH1A1TSHRLMNAMAPTDPP4
SCHEMBL4668963 0.87 DPP4 (0.78) ALDH1A1TSHRLMNAMAPTDPP4
SCHEMBL8337418 0.87 ALDH1A1 (0.74) ALDH1A1NPSR1TSHRLMNAHTT
SCHEMBL13939265 0.86 DPP4 (0.81) ALDH1A1NPSR1TSHRLMNAHTT
SCHEMBL12604413 0.86 DPP4 (0.81) ALDH1A1NPSR1TSHRLMNAHTT
SCHEMBL4668737 0.85 DPP4 (0.71) ALDH1A1NPSR1TSHRLMNAHTT
SCHEMBL4076753 0.85 DPP4 (0.71) ALDH1A1NPSR1TSHRLMNAHTT
SCHEMBL4668639 0.85 DPP4 (0.71) ALDH1A1NPSR1TSHRLMNAHTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2003057200-A2 COMPOSITIONS COMPRISING INHIBITORS OF DPP-IV AND NEP ENZYMES FOR THE TREATMENT OF DIABETES NOVO NORDISK A/S (DK) 2003-07-17 WO disclosed
WO-2003004496-A1 DPP-IV-INHIBITING PURINE DERIVATIVES FOR THE TREATMENT OF DIABETES NOVO NORDISK A/S (DK) 2003-01-16 WO disclosed