SCHEMBL8353178

SCHEMBL8353178

Cc1ccc(C2(CCNC3CC3)CC2)cc1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 1/20 0.42
OPRM1 P35372 3/20 0.41
LMNA P02545 3/20 0.38
ALDH1A1 P00352 3/20 0.38
NPSR1 Q6W5P4 3/20 0.38
SMN1; SMN2 Q16637 2/20 0.38
GAA P10253 1/20 0.38
ICMT O60725 3/20 0.36
SLC6A2 P23975 1/20 0.36
SLC6A4 P31645 1/20 0.36
SLC6A3 Q01959 1/20 0.36
CYP3A4 P08684 1/20 0.36
CYP2D6 P10635 1/20 0.36
CYP2C9 P11712 1/20 0.36
CYP2C19 P33261 1/20 0.36
HTT P42858 1/20 0.36
HTR1A P08908 1/20 0.36
HTR7 P34969 1/20 0.36
HTR6 P50406 1/20 0.36
MEN1 O00255 2/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8353652 0.94 KDM4E (0.43) KDM4EOPRM1LMNAALDH1A1NPSR1
SCHEMBL14347879 0.94 SLC6A4 (0.43) KDM4EOPRM1LMNAALDH1A1NPSR1
SCHEMBL8353273 0.83 SLC6A4 (0.51) KDM4ELMNASMN1; SMN2SLC6A2SLC6A4
SCHEMBL14347818 0.79 OPRM1 (0.45) OPRM1LMNAALDH1A1NPSR1SMN1; SMN2
SCHEMBL8350796 0.77 SLC6A4 (0.60) KDM4ELMNANPSR1SMN1; SMN2SLC6A2
SCHEMBL8353275 0.77 SLC6A4 (0.49) KDM4ELMNAALDH1A1SMN1; SMN2SLC6A2
SCHEMBL8353030 0.77 SLC6A4 (0.49) KDM4ELMNAALDH1A1SMN1; SMN2SLC6A2
Hydrochloric Acid SCHEMBL11113043 0.76 SLC6A4 (0.46) OPRM1LMNAALDH1A1NPSR1SLC6A2
SCHEMBL8353624 0.75 SMN1; SMN2 (0.43) OPRM1LMNAALDH1A1NPSR1SMN1; SMN2
SCHEMBL8355218 0.73 OPRM1 (0.50) OPRM1LMNAALDH1A1NPSR1SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7312214-B2 1, 1-disubstituted cycloalkyl derivatives as factor Xa inhibitors BRISTOL-MYERS SQUIBB COMPANY (US) 2007-12-25 US disclosed
WO-2003099276-A1 1,1-DISUBSTITUTED CYCLOALKYL DERIVATIVES AS FACTOR XA INHIBITORS BRISTOL-MYERS SQUIBB COMPANY (US) 2003-12-04 WO disclosed