SCHEMBL8353448

SCHEMBL8353448

COCCN1CC(C)CN(CCOC)C1

nearest known ligand 0.46

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
GBA1 P04062 2/20 0.46
ALDH1A1 P00352 2/20 0.35
HSD11B1 P28845 1/20 0.33
CYP2D6 P10635 1/20 0.33
SLC6A2 P23975 1/20 0.33
SLC6A4 P31645 1/20 0.33
SLC6A3 Q01959 1/20 0.33
KCNH2 Q12809 1/20 0.33
KDM4E B2RXH2 2/20 0.32
MEN1 O00255 1/20 0.32
KMT2A Q03164 1/20 0.32
SMN1; SMN2 Q16637 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18484868 0.91
SCHEMBL24461055 0.83 GBA1 (0.47) GBA1ALDH1A1HSD11B1KDM4EMEN1
SCHEMBL2844152 0.80 GBA1 (0.41) GBA1ALDH1A1HSD11B1CYP2D6SLC6A2
SCHEMBL497158 0.79 GBA1 (0.38) GBA1ALDH1A1HSD11B1CYP2D6SLC6A2
SCHEMBL12449698 0.78 ALDH1A1 (0.46) GBA1ALDH1A1CYP2D6KDM4E
SCHEMBL12951 0.78 ALDH1A1 (0.46) GBA1ALDH1A1CYP2D6KDM4E
SCHEMBL12449700 0.78 ALDH1A1 (0.46) GBA1ALDH1A1CYP2D6KDM4E
SCHEMBL19938007 0.76 GBA1 (0.48) GBA1ALDH1A1HSD11B1CYP2D6SLC6A2
SCHEMBL12449655 0.75 KDM4E (0.55) ALDH1A1KDM4EKMT2A
SCHEMBL12837 0.75 KDM4E (0.55) ALDH1A1KDM4EKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7629468-B2 Neuroprotectants, analgesics or anticonvulsants JANSSEN PHARMACEUTICA NV (BE) 2009-12-08 US disclosed
US-7629468-B2 Neuroprotectants, analgesics or anticonvulsants JANSSEN PHARMACEUTICA NV (BE) 2009-12-08 US disclosed
US-7517517-B2 Radiolabelled quinoline and quinolinone derivatives and their use as metabotropic glutamate receptor ligands JANSSEN PHARMACEUTICA N.V. (BE) 2009-04-14 US disclosed
US-7517517-B2 Radiolabelled quinoline and quinolinone derivatives and their use as metabotropic glutamate receptor ligands JANSSEN PHARMACEUTICA N.V. (BE) 2009-04-14 US disclosed
WO-2003082350-A2 RADIOLABELLED QUINOLINE AND QUINOLINONE DERIVATIVES AND THEIR USE AS METABOTROPIC GLUTAMATE RECEPTOR LIGANDS JANSSEN PHARMACEUTICA N.V. (BE) 2003-10-09 WO disclosed