SCHEMBL8353945

SCHEMBL8353945

Cc1ccc(C2(CN3CCOCC3)CCC2)cc1

nearest known ligand 0.58

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
SLC6A2 P23975 4/20 0.58
SLC6A4 P31645 4/20 0.58
SLC6A3 Q01959 3/20 0.58
POLB P06746 2/20 0.40
HSD11B1 P28845 1/20 0.39
MAPK1 P28482 1/20 0.39
NPC1 O15118 1/20 0.39
RAB9A P51151 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.39
MEN1 O00255 1/20 0.38
CYP3A4 P08684 1/20 0.38
TSHR P16473 1/20 0.38
CYP2C19 P33261 1/20 0.38
KMT2A Q03164 1/20 0.38
FAAH O00519 1/20 0.38
ALDH1A1 P00352 1/20 0.38
MGLL Q99685 1/20 0.38
FPR2 P25090 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8351474 0.97 SLC6A2 (0.62) SLC6A2SLC6A4SLC6A3POLBHSD11B1
SCHEMBL12386 0.94 SLC6A2 (0.54) SLC6A2SLC6A4SLC6A3POLBHSD11B1
SCHEMBL8353033 0.87 SLC6A2 (0.54) SLC6A2SLC6A4SLC6A3HSD11B1MEN1
SCHEMBL8355835 0.85 POLB (0.45) SLC6A2SLC6A4SLC6A3POLBRAB9A
SCHEMBL8351046 0.83 SLC6A2 (0.58) SLC6A2SLC6A4SLC6A3HSD11B1MEN1
SCHEMBL8351497 0.82 SLC6A2 (0.46) SLC6A2SLC6A4SLC6A3POLBRAB9A
SCHEMBL8352677 0.82 SLC6A2 (0.51) SLC6A2SLC6A4SLC6A3HSD11B1ALDH1A1
SCHEMBL8352799 0.78 POLB (0.47) POLBRAB9ASMN1; SMN2TSHRALDH1A1
SCHEMBL10640 0.78 SLC6A2 (0.54) SLC6A2SLC6A4SLC6A3HSD11B1FPR2
SCHEMBL17080540 0.78 SLC6A2 (0.54) SLC6A2SLC6A4SLC6A3HSD11B1NPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7312214-B2 1, 1-disubstituted cycloalkyl derivatives as factor Xa inhibitors BRISTOL-MYERS SQUIBB COMPANY (US) 2007-12-25 US disclosed
WO-2003099276-A1 1,1-DISUBSTITUTED CYCLOALKYL DERIVATIVES AS FACTOR XA INHIBITORS BRISTOL-MYERS SQUIBB COMPANY (US) 2003-12-04 WO disclosed