SCHEMBL8354909

SCHEMBL8354909

COC(=O)[C@@H]1C[C@@H](Oc2cc(-c3ccccc3)nc3cc(OC)ccc23)CN1C(=O)[C@@H](NC(=O)OC(C)(C)C)C(C)(C)C

nearest known ligand 0.49

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 1/20 0.45
KDM4E B2RXH2 1/20 0.42
ALDH1A1 P00352 1/20 0.42
SMN1; SMN2 Q16637 1/20 0.42
ELANE P08246 7/20 0.42
TACR3 P29371 6/20 0.41
PLA2G2A P14555 1/20 0.38
CTSB P07858 1/20 0.38
PPP3CB P16298 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4981257 1.00 CYP3A4 (0.45) CYP3A4KDM4EALDH1A1SMN1; SMN2ELANE
Corboxylic Acid SCHEMBL8273022 0.95 CYP3A4 (0.46) CYP3A4KDM4EALDH1A1SMN1; SMN2ELANE
Corboxylic Acid SCHEMBL5692528 0.95 CYP3A4 (0.46) CYP3A4KDM4EALDH1A1SMN1; SMN2ELANE
Corboxylic Acid SCHEMBL13997824 0.95 CYP3A4 (0.46) CYP3A4KDM4EALDH1A1SMN1; SMN2ELANE
Corboxylic Acid SCHEMBL30966182 0.95 CYP3A4 (0.46) CYP3A4KDM4EALDH1A1SMN1; SMN2ELANE
SCHEMBL5692538 0.92 KDM4E (0.42) CYP3A4KDM4EALDH1A1SMN1; SMN2ELANE
SCHEMBL8275068 0.91 CTSB (0.46) CYP3A4KDM4EALDH1A1SMN1; SMN2TACR3
SCHEMBL8355920 0.91 KDM4E (0.43) CYP3A4KDM4EALDH1A1SMN1; SMN2ELANE
SCHEMBL8353025 0.90 CYP3A4 (0.50) CYP3A4KDM4EALDH1A1SMN1; SMN2ELANE
SCHEMBL8354706 0.89 CYP3A4 (0.48) CYP3A4KDM4EALDH1A1SMN1; SMN2ELANE

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2004043339-A2 SUBSTITUTED CYCLOALKYL P1' HEPATITIS C VIRUS INHIBITORS BRISTOL-MYERS SQUIBB COMPANY (US) 2004-05-27 WO disclosed