SCHEMBL8355083

SCHEMBL8355083

O=[N+]([O-])c1cccc(-c2csc(NS(=O)(=O)c3ccc(Cl)cc3)n2)c1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
KDM1A O60341 11/20 0.84
KMO O15229 1/20 0.70
MAOA P21397 4/20 0.69
MEN1 O00255 1/20 0.69
POLB P06746 1/20 0.69
KMT2A Q03164 1/20 0.69

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3673316 0.91 KDM1A (0.80) KDM1AKMOMAOAMEN1POLB
SCHEMBL2762558 0.90 MEN1 (0.77) KDM1AKMOMAOAMEN1POLB
SCHEMBL8359357 0.89 KDM1A (0.81) KDM1AKMOMAOAMEN1POLB
SCHEMBL727088 0.89 KDM1A (0.74) KDM1AKMOMAOAMEN1POLB
SCHEMBL728110 0.89 KDM1A (0.74) KDM1AKMOMAOAMEN1POLB
SCHEMBL8360638 0.89 KDM1A (0.73) KDM1AKMOMAOAMEN1POLB
SCHEMBL2762772 0.88 KDM1A (0.76) KDM1AKMOMAOAMEN1POLB
SCHEMBL726766 0.86 KMO (0.79) KDM1AKMOMAOAMEN1POLB
SCHEMBL2762482 0.85 KDM1A (0.68) KDM1AKMOMAOAMEN1POLB
SCHEMBL2762510 0.84 KDM1A (0.69) KDM1AKMOMAOAMEN1POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5877193-A NERVOUS SYSTEM DISORDERS; PSYCHOLOGICAL DISORDERS HOFFMANN-LA ROCHE INC. (US) 1999-03-02 US claimed
US-5958910-A Use of N-(4-aryl-thiazol-2-yl)-sulfonamides HOFFMANN-LA ROCHE INC. (US) 1999-09-28 US disclosed
US-5877193-A NERVOUS SYSTEM DISORDERS; PSYCHOLOGICAL DISORDERS HOFFMANN-LA ROCHE INC. (US) 1999-03-02 US disclosed
EP-0819681-A2 N-(4-Aryl-thiazol-2-yl)-sulfonamides and their use F. HOFFMANN-LA ROCHE AG (CH) 1998-01-21 EP disclosed