SCHEMBL8356014

SCHEMBL8356014

COc1ccc(-c2cc(=O)c3c(O)cc(OCC(=O)N(C)C)cc3o2)cc1OC1CC2CCC2C1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1B1 Q16678 4/20 0.53
CYP1A1 P04798 3/20 0.51
CYP1A2 P05177 2/20 0.51
ABCC1 P33527 2/20 0.51
KDM1A O60341 2/20 0.51
HDAC6 Q9UBN7 2/20 0.51
IP6K2 Q9UHH9 2/20 0.51
XDH P47989 2/20 0.51
IPMK Q8NFU5 1/20 0.51
PPARG P37231 1/20 0.50
MEN1 O00255 1/20 0.48
ALDH1A1 P00352 1/20 0.48
POLB P06746 1/20 0.48
MAPT P10636 1/20 0.48
KMT2A Q03164 1/20 0.48
PLG P00747 1/20 0.48
EPHX2 P34913 1/20 0.47
FLT3 P36888 1/20 0.45
MKNK2 Q9HBH9 1/20 0.45
CYP19A1 P11511 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7310036 0.92 CYP1B1 (0.55) CYP1B1CYP1A1CYP1A2ABCC1KDM1A
SCHEMBL7303648 0.90 CYP1B1 (0.51) CYP1B1CYP1A1CYP1A2ABCC1KDM1A
SCHEMBL7304881 0.85 CYP1B1 (0.53) CYP1B1CYP1A1CYP1A2ABCC1KDM1A
SCHEMBL7307391 0.84 CYP1B1 (0.53) CYP1B1CYP1A1CYP1A2ABCC1KDM1A
SCHEMBL7309697 0.83 CYP1B1 (0.58) CYP1B1CYP1A1CYP1A2ABCC1KDM1A
SCHEMBL7303645 0.82 CYP1B1 (0.57) CYP1B1CYP1A1CYP1A2ABCC1KDM1A
SCHEMBL7311118 0.82 CYP1B1 (0.57) CYP1B1CYP1A1CYP1A2ABCC1KDM1A
SCHEMBL7316873 0.82 CYP1B1 (0.57) CYP1B1CYP1A1CYP1A2ABCC1KDM1A
SCHEMBL8327175 0.82 CYP3A4 (0.42) CYP1A2MEN1ALDH1A1POLBMAPT
SCHEMBL7318625 0.82 CYP1B1 (0.56) CYP1B1CYP1A1CYP1A2ABCC1KDM1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2003024488-A2 COMBINATION OF A PDE INHIBITOR AND A LEUKOTRIENE RECEPTOR ANTAGONIST ALTANA PHARMA AG (DE) 2003-03-27 WO disclosed