SCHEMBL8357

SCHEMBL8357

O=C(O)[C@H]1NCCS1

nearest known ligand 0.00

⚠ Novel chemotype — no close known analogue (best Tanimoto < 0.3). Unexplored chemical space relative to ChEMBL.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2030154 1.00
SCHEMBL23170 1.00
SCHEMBL29818313 0.98
Hydrochloric Acid SCHEMBL16798191 0.98
Hydrochloric Acid SCHEMBL202670 0.98
Formic Acid SCHEMBL6596895 0.91 SLC1A2 (0.33)
SCHEMBL5293023 0.86
Pipecolic Acid SCHEMBL8894672 0.83 DPP4 (0.41)
SCHEMBL23421623 0.82 MAPT (0.32)
SCHEMBL2532769 0.82 MAPT (0.32)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Appears in 3433 patents — a generic fragment claimed broadly, so it's down-weighted as IP noise. Top by claim status then date:

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20260091067-A1 METHODS AND USES OF MICROBIOME COMPOSITIONS, COMPONENTS, OR METABOLITES FOR TREATING INSULIN-ASSOCIATED DISEASES MARVELBIOME INC (US) 2026-04-02 US claimed
EP-4679087-A1 BIOMARKER AND USE THEREOF MEIJI CO., LTD (JP) 2026-01-14 EP claimed
US-20250361490-A1 COMPOSITION AND METHOD FOR CRYOPRESERVATION OF MITOCHONDRIA CELLVIE AG (CH) 2025-11-27 US claimed
US-12428447-B2 Peptide-based non-proteinaceous cargo delivery FELDAN BIO INC. (CA) 2025-09-30 US claimed
EP-4587116-A2 METHODS AND USES OF MICROBIOME COMPOSITIONS, COMPONENTS, OR METABOLITES FOR TREATING INSULIN-ASSOCIATED DISEASES MarvelBiome, Inc. (US) 2025-07-23 EP claimed
EP-4535996-A1 COMPOSITION AND METHOD FOR CRYOPRESERVATION OF MITOCHONDRIA cellvie AG (CH) 2025-04-16 EP claimed
WO-2025054048-A1 METHODS AND USES OF MICROBIOME COMPOSITIONS, COMPONENTS, OR METABOLITES FOR TREATING LIPID AND CHOLESTEROL METABOLISM ASSOCIATED DISEASES, DISORDERS, AND CONDITIONS MarvelBiome, Inc. (US) 2025-03-13 WO claimed
WO-2025032025-A1 STABLE GLASSY MATERIAL BASED ON HISTIDINE, ARGININE AND GLUTAMIC ACID AMINO ACIDS VITROPEP (FR) 2025-02-13 WO claimed
CN-119365073-A Compositions and methods for cryopreserving mitochondria 赛立维公司 2025-01-24 CN claimed
EP-4440342-A1 METHODS AND USES OF MICROBIOME COMPOSITIONS, COMPONENTS, OR METABOLITES FOR TREATING VAGUS NERVE ASSOCIATED DISEASES, DISORDERS, AND CONDITIONS MarvelBiome, Inc. (US) 2024-10-09 EP claimed
WO-2005112999-A2 CANCER TREATMENT WITH INHIBITORS OF COLLAGEN SYNTHESIS VECTRAMED, INC. (US) 2005-12-01 WO claimed
US-20050118180-A1 Inhibition of abnormal cell proliferation with camptothecin and combinations including the same SUPERGEN, INC. 2005-06-02 US claimed
EP-1276479-A2 INHIBITION OF ABNORMAL CELL PROLIFERATION WITH CAMPTOTHECIN AND COMBINATIONS INCLUDING THE SAME SuperGen, Inc. (US) 2003-01-22 EP claimed
US-20020111362-A1 Inhibition of abnormal cell proliferation with camptothecin and combinations including the same SUPERGEN, INC. 2002-08-15 US claimed
WO-2001080843-A2 INHIBITION OF ABNORMAL CELL PROLIFERATION WITH CAMPTOTHECIN AND COMBINATIONS INCLUDING THE SAME SUPERGEN, INC. (US) 2001-11-01 WO claimed
US-6251249-B1 IODIDE-FREE AND CONTAIN AN ORGANOSULFUR COMPOUND AND/OR A CARBOXYLIC ACID; PRECIOUS METAL ALKANESULFONATES, PRECIOUS METAL ALKANESULFONAMIDES AND/OR PRECIOUS METAL SOURCE ATOFINA CHEMICALS, INC. 2001-06-26 US claimed
EP-0672678-B1 Azapeptide derivative FUJIREBIO KK (JP) 2000-10-25 EP claimed
US-5965538-A FOR TREATING NERVOUS INFLAMMATION OF RESPIRATORY SYSTEMS, ASTHMA, BRONCHOSPASM FUJIREBIO INC. (JP) 1999-10-12 US claimed
US-5770574-A Long-chain alkylamides of amino acids and peptides with anti-proliferative and anti-inflammatory properties ASTA MEDICA AKTIENGESELLSCHAFT (DE) 1998-06-23 US claimed
EP-0672678-A1 Azapeptide derivative FUJIREBIO Inc. (JP) 1995-09-20 EP claimed