SCHEMBL8358016

SCHEMBL8358016

CCOc1ccc2nc(NC(=O)CBr)sc2c1.O=C(Br)CBr

nearest known ligand 0.73

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 7/20 0.73
NPC1 O15118 5/20 0.73
RAB9A P51151 5/20 0.73
HSD17B10 Q99714 1/20 0.73
TP53 P04637 2/20 0.72
MAPK1 P28482 2/20 0.72
POLB P06746 2/20 0.72
ALDH1A1 P00352 1/20 0.72
HTT P42858 1/20 0.72
CSNK1D P48730 7/20 0.67
P2RY12 Q9H244 1/20 0.67
MAPT P10636 6/20 0.64
CASP3 P42574 1/20 0.64
SENP8 Q96LD8 1/20 0.64
SENP7 Q9BQF6 1/20 0.64
SENP6 Q9GZR1 1/20 0.64
GAA P10253 1/20 0.63
SIRT2 Q8IXJ6 1/20 0.63
MEN1 O00255 1/20 0.63
USP2 O75604 1/20 0.63

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8353831 0.96 SMN1; SMN2 (0.78) SMN1; SMN2NPC1RAB9AHSD17B10TP53
SCHEMBL8350055 0.88 CASP2 (0.72) SMN1; SMN2NPC1RAB9ATP53ALDH1A1
SCHEMBL6229213 0.87 SMN1; SMN2 (0.82) SMN1; SMN2NPC1RAB9AHSD17B10TP53
SCHEMBL10576093 0.85 SMN1; SMN2 (0.78) SMN1; SMN2NPC1RAB9AHSD17B10TP53
SCHEMBL14202814 0.85 SMN1; SMN2 (0.78) SMN1; SMN2NPC1RAB9AHSD17B10TP53
SCHEMBL27022345 0.85 SMN1; SMN2 (0.78) SMN1; SMN2NPC1RAB9AHSD17B10TP53
SCHEMBL29500248 0.84 CASP2 (0.77) SMN1; SMN2NPC1RAB9ATP53ALDH1A1
SCHEMBL8353964 0.84 CASP2 (0.77) SMN1; SMN2NPC1RAB9ATP53ALDH1A1
SCHEMBL9332424 0.84 SMN1; SMN2 (1.00) SMN1; SMN2NPC1RAB9AHSD17B10TP53
SCHEMBL15376318 0.83 MAPT (0.78) SMN1; SMN2NPC1RAB9AHSD17B10TP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1999031096-A1 PIPERAZINE DERIVATIVES USEFUL AS HYPOGLYCEMIC AGENTS SHAMAN PHARMACEUTICALS, INC. (US) 1999-06-24 WO disclosed