SCHEMBL8359484

SCHEMBL8359484

NCC(=O)N1CCc2[nH]c(=O)c3ccccc3c2C1

nearest known ligand 0.71

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 14/20 0.71
TAAR1 Q96RJ0 1/20 0.53
MAPT P10636 2/20 0.51
LMNA P02545 1/20 0.51
BAZ2B Q9UIF8 1/20 0.51
GAA P10253 1/20 0.49
ALDH1A1 P00352 2/20 0.48
CASP1 P29466 2/20 0.48
CASP7 P55210 2/20 0.48
KDM4E B2RXH2 1/20 0.48
MEN1 O00255 1/20 0.47
ALOX15 P16050 1/20 0.47
KMT2A Q03164 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8359597 0.91 PARP1 (0.74) PARP1TAAR1MAPTLMNABAZ2B
SCHEMBL8360520 0.90 PARP1 (0.71) PARP1
SCHEMBL14444059 0.87 PARP1 (0.71) PARP1TAAR1MAPTLMNABAZ2B
SCHEMBL14444062 0.86 PARP1 (0.73) PARP1TAAR1MAPTLMNABAZ2B
SCHEMBL8359333 0.85 PARP1 (0.72) PARP1TAAR1MAPTLMNABAZ2B
SCHEMBL8363074 0.84 PARP1 (0.67) PARP1TAAR1MAPTLMNABAZ2B
SCHEMBL8363089 0.83 PARP1 (1.00) PARP1MAPTGAAALDH1A1CASP1
SCHEMBL14444067 0.83 PARP1 (0.73) PARP1TAAR1MAPTLMNABAZ2B
SCHEMBL8363073 0.83 PARP1 (0.83) PARP1MAPTGAAALDH1A1CASP1
SCHEMBL8359275 0.83 BAZ2B (0.73) PARP1MAPTLMNABAZ2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7247641-B2 Compounds, derivatives, compositions, preparation and uses MGI GP, INC. (US) 2007-07-24 US disclosed
US-7247641-B2 Compounds, derivatives, compositions, preparation and uses MGI GP, INC. (US) 2007-07-24 US disclosed
WO-2003014121-A9 COMPOUNDS, DERIVATIVES, COMPOSITIONS, PREPARATION AND USES GUILFORD PHARM INC (US) 2004-03-25 WO disclosed
WO-2003014121-A1 COMPOUNDS, DERIVATIVES, COMPOSITIONS, PREPARATION AND USES GUILFORD PHARMACEUTICALS INC. (US) 2003-02-20 WO disclosed