SCHEMBL8360520

SCHEMBL8360520

NCC(=O)N1CCc2c([nH]c(=O)c3ccccc23)C1

nearest known ligand 0.71

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 13/20 0.71
GPX4 P36969 1/20 0.57
HDAC6 Q9UBN7 3/20 0.49
HDAC1 Q13547 2/20 0.49
FAAH O00519 1/20 0.46
TRPV1 Q8NER1 1/20 0.46
CDK4 P11802 1/20 0.46
CCND1 P24385 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8360521 0.91 PARP1 (0.73) PARP1GPX4HDAC6HDAC1TRPV1
SCHEMBL8359484 0.90 PARP1 (0.71) PARP1
SCHEMBL5556447 0.86 GPX4 (0.77) GPX4HDAC6HDAC1FAAHTRPV1
SCHEMBL8359246 0.85 PARP1 (0.68) PARP1GPX4HDAC6HDAC1TRPV1
SCHEMBL8363099 0.84 PARP1 (0.67) PARP1GPX4HDAC6HDAC1FAAH
SCHEMBL5367984 0.84 PARP1 (0.66) PARP1GPX4FAAHTRPV1CDK4
SCHEMBL30023116 0.84 PARP1 (0.66) PARP1GPX4FAAHTRPV1CDK4
SCHEMBL8360509 0.83 PARP1 (0.69) PARP1GPX4HDAC6HDAC1TRPV1
SCHEMBL8363098 0.83 PARP1 (1.00) PARP1GPX4
SCHEMBL8363110 0.82 PARP1 (0.61) PARP1GPX4HDAC6HDAC1CDK4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7247641-B2 Compounds, derivatives, compositions, preparation and uses MGI GP, INC. (US) 2007-07-24 US disclosed
US-7247641-B2 Compounds, derivatives, compositions, preparation and uses MGI GP, INC. (US) 2007-07-24 US disclosed
WO-2003014121-A9 COMPOUNDS, DERIVATIVES, COMPOSITIONS, PREPARATION AND USES GUILFORD PHARM INC (US) 2004-03-25 WO disclosed
WO-2003014121-A1 COMPOUNDS, DERIVATIVES, COMPOSITIONS, PREPARATION AND USES GUILFORD PHARMACEUTICALS INC. (US) 2003-02-20 WO disclosed