SCHEMBL836061

SCHEMBL836061

Cc1ccc(Sc2cc(=O)n(C)c3cc(Cl)ccc23)cc1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.54
CYP3A4 P08684 2/20 0.54
CYP2C19 P33261 2/20 0.54
CYP1A2 P05177 1/20 0.54
CYP2C9 P11712 1/20 0.54
ALOX15 P16050 1/20 0.54
TSHR P16473 1/20 0.54
HSD17B10 Q99714 1/20 0.54
NPSR1 Q6W5P4 3/20 0.50
HPGD P15428 3/20 0.50
RHEB Q15382 1/20 0.50
KDM4E B2RXH2 6/20 0.47
SMN1; SMN2 Q16637 2/20 0.47
MAPT P10636 3/20 0.47
ENPP2 Q13822 1/20 0.44
L3MBTL1 Q9Y468 2/20 0.43
TP53 P04637 2/20 0.43
AKR1B1 P15121 1/20 0.43
PTGDR2 Q9Y5Y4 1/20 0.43
POLB P06746 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL835025 0.88 ALDH1A1 (0.50) ALDH1A1CYP3A4CYP2C19CYP1A2CYP2C9
SCHEMBL836059 0.84 RHEB (0.50) ALDH1A1CYP2C9ALOX15TSHRNPSR1
SCHEMBL14300144 0.83 RXFP1 (0.58) ALDH1A1TSHRHSD17B10NPSR1HPGD
SCHEMBL835184 0.82 KDM4E (0.58) ALDH1A1CYP3A4CYP2C19CYP1A2CYP2C9
SCHEMBL835232 0.82 KDM4E (0.44) ALDH1A1CYP3A4CYP2C19CYP1A2CYP2C9
SCHEMBL836066 0.80 RXFP1 (0.48) ALDH1A1HSD17B10NPSR1HPGDRHEB
SCHEMBL836042 0.77 HTT (0.49) ALDH1A1CYP3A4CYP2C19CYP1A2CYP2C9
SCHEMBL835001 0.76 RXFP1 (0.44) ALDH1A1HSD17B10NPSR1RHEBKDM4E
SCHEMBL835197 0.75 RXFP1 (0.49) ALDH1A1CYP3A4CYP2C19CYP1A2ALOX15
SCHEMBL30901294 0.75 NQO2 (0.61) ALDH1A1CYP3A4CYP2C19CYP1A2CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8143276-B2 4-thio substituted quinoline and naphthyridine compounds XTL BIOPHARMACEUTICALS LTD. (IL) 2012-03-27 US disclosed