SCHEMBL8360874

SCHEMBL8360874

CCOC(=O)c1cc(-c2cnc(NC(C)C)c(=O)n2CC(=O)O)cc([N+](=O)[O-])c1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
F7 P08709 11/20 0.42
NPC1 O15118 2/20 0.42
F3 P13726 2/20 0.41
FOS P01100 1/20 0.39
JUN P05412 1/20 0.39
NFKB1 P19838 1/20 0.39
NFKB2 Q00653 1/20 0.39
RELA Q04206 1/20 0.39
MAPT P10636 3/20 0.37
KDM4E B2RXH2 1/20 0.37
RAB9A P51151 1/20 0.37
POLB P06746 1/20 0.36
DYRK3 O43781 1/20 0.35
CCNT1 O60563 1/20 0.35
CCNA2 P20248 1/20 0.35
CDK2 P24941 1/20 0.35
CDK9 P50750 1/20 0.35
CDK5 Q00535 1/20 0.35
DYRK1A Q13627 1/20 0.35
CDK5R1 Q15078 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6791732 0.88 F7 (0.48) F7F3
SCHEMBL6791726 0.88 F7 (0.48) F7F3
SCHEMBL8362430 0.86 F7 (0.56) F7NPC1F3DYRK3CCNT1
SCHEMBL8360867 0.85 F7 (0.42) F7F3MAPTGAA
SCHEMBL6794526 0.85 F7 (0.44) F7F3MAPTGAA
SCHEMBL8360872 0.85 F7 (0.43) F7F3MAPTKDM4EGAA
SCHEMBL6794515 0.85 F7 (0.44) F7F3MAPTGAA
SCHEMBL6797477 0.84 F7 (0.43) F7F3GAA
SCHEMBL6797466 0.84 F7 (0.43) F7F3GAA
SCHEMBL6794077 0.83 F7 (0.44) F7NPC1F3FOSJUN

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2003028729-A2 PRODRUGS OF SUBSTITUTED POLYCYCLIC COMPOUNDS USEFUL FOR SELECTIVE INHIBITION OF THE COAGULATION CASCADE PHARMACIA CORPORATION (US) 2003-04-10 WO disclosed