SCHEMBL8362000

SCHEMBL8362000

Clc1ccc(CSc2nc3ccc(OCCN4CCCCC4)cc3s2)cc1

nearest known ligand 0.57

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 1/20 0.57
TSHR P16473 1/20 0.57
RAB9A P51151 1/20 0.57
MAPT P10636 3/20 0.53
L3MBTL1 Q9Y468 2/20 0.53
LMNA P02545 1/20 0.53
MAPK1 P28482 1/20 0.53
HTT P42858 1/20 0.53
TDP1 Q9NUW8 1/20 0.53
LTA4H P09960 6/20 0.51
TMEM97 Q5BJF2 2/20 0.50
AURKB Q96GD4 3/20 0.48
PTGS2 P35354 1/20 0.47
ACHE P22303 2/20 0.47
HRH3 Q9Y5N1 2/20 0.46
POLB P06746 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8361504 0.99 NPC1 (0.55) NPC1TSHRRAB9AMAPTL3MBTL1
SCHEMBL8359521 0.83 LTA4H (0.60) NPC1TSHRRAB9ALTA4HAURKB
SCHEMBL8357943 0.82 MAPT (0.60) NPC1RAB9AMAPTL3MBTL1LMNA
SCHEMBL8362101 0.82 LTA4H (0.61) NPC1TSHRRAB9ALTA4HAURKB
SCHEMBL8358459 0.81 MAPT (0.58) NPC1RAB9AMAPTL3MBTL1LMNA
SCHEMBL8361623 0.80 MAPT (0.80) NPC1TSHRRAB9AMAPTL3MBTL1
SCHEMBL8355863 0.80 MAPT (0.60) NPC1RAB9AMAPTL3MBTL1LMNA
SCHEMBL8359745 0.80 MAPT (0.60) NPC1RAB9AMAPTL3MBTL1LMNA
SCHEMBL8355890 0.78 MAPT (0.61) NPC1RAB9AMAPTL3MBTL1LMNA
SCHEMBL8361935 0.77 MAPT (0.60) NPC1RAB9AMAPTL3MBTL1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5919807-A ANTICHOLESTEROL AGENTS DR. KARL THOMAE GMBH (DE) 1999-07-06 US disclosed
EP-0824529-A1 BENZOTHIAZOLES AND BENZOXAZOLES, AS WELL AS DRUGS CONTAINING THEM, THEIR USE AND METHODS OF PREPARING THEM Dr. Karl Thomae GmbH (DE) 1998-02-25 EP disclosed
WO-1996035681-A1 BENZOTHIAZOLES AND BENZOXAZOLES, AS WELL AS DRUGS CONTAINING THEM, THEIR USE AND METHODS OF PREPARING THEM DR. KARL THOMAE GMBH (DE) 1996-11-14 WO disclosed