SCHEMBL8364101

SCHEMBL8364101

CS(=O)(=O)CCN(CCCCOc1ccc2ncnc(Nc3ccc(OCc4cccc(F)c4)c(Cl)c3)c2c1)C(=O)C(F)(F)F

nearest known ligand 0.74

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ERBB2 P04626 17/20 0.74
EGFR P00533 17/20 0.74
MEN1 O00255 3/20 0.56
KMT2A Q03164 3/20 0.56
ERBB4 Q15303 2/20 0.56
CYP3A4 P08684 2/20 0.56
PIK3C2B O00750 1/20 0.56
MAP2K7 O14733 1/20 0.56
RIPK2 O43353 1/20 0.56
PIK3C2G O75747 1/20 0.56
STK10 O94804 1/20 0.56
ABCB11 O95342 1/20 0.56
ABL1 P00519 1/20 0.56
INSR P06213 1/20 0.56
RET P07949 1/20 0.56
PDGFRB P09619 1/20 0.56
SRC P12931 1/20 0.56
CYP3A5 P20815 1/20 0.56
ERBB3 P21860 1/20 0.56
CDK2 P24941 1/20 0.56

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6954812 0.89 EGFR (0.59) ERBB2EGFRMEN1KMT2AERBB4
SCHEMBL8365368 0.85 EGFR (1.00) ERBB2EGFRERBB4AURKB
SCHEMBL8366002 0.84 EGFR (1.00) ERBB2EGFRMEN1KMT2AERBB4
SCHEMBL16180163 0.84 EGFR (0.79) ERBB2EGFRMEN1KMT2AERBB4
SCHEMBL3697748 0.81 EGFR (0.49) ERBB2EGFRALDH1A1
SCHEMBL2505727 0.81 ERBB2 (0.75) ERBB2EGFRERBB4ABL1INSR
SCHEMBL4335805 0.79 EGFR (0.78) ERBB2EGFRERBB4ABL1INSR
SCHEMBL4348156 0.79 ERBB2 (0.68) ERBB2EGFRERBB4ABL1INSR
SCHEMBL8367168 0.79 EGFR (0.89) ERBB2EGFRMEN1KMT2AERBB4
SCHEMBL12200048 0.79 ERBB2 (0.75) ERBB2EGFRERBB4ABL1INSR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1999035132-A1 HETEROCYCLIC COMPOUNDS GLAXO GROUP LIMITED (GB) 1999-07-15 WO disclosed