SCHEMBL8364502

SCHEMBL8364502

CCOC(=O)c1c(C)n(-c2ccc(-c3ccccc3-c3noc(C(Cl)(Cl)Cl)n3)cc2)c2sc(CC)cc2c1=O

nearest known ligand 0.37

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
AGTR1 P30556 10/20 0.37
THRB P10828 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
TP53 P04637 1/20 0.34
KDM4E B2RXH2 1/20 0.34
ALDH1A1 P00352 1/20 0.34
HPGD P15428 1/20 0.34
GRM6 O15303 1/20 0.34
MAPT P10636 2/20 0.34
MEN1 O00255 1/20 0.34
KMT2A Q03164 1/20 0.34
AR P10275 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7010779 0.81 AGTR1 (0.41) AGTR1
SCHEMBL8362047 0.80 CHEK1 (0.39) AGTR1THRBSMN1; SMN2KDM4EALDH1A1
SCHEMBL2775939 0.71 AGTR1 (0.50) AGTR1
SCHEMBL8359936 0.68 AGTR1 (0.45) AGTR1KDM4EALDH1A1HPGD
SCHEMBL8363467 0.67 AGTR1 (0.36) AGTR1
SCHEMBL7014100 0.67 AGTR1 (0.46) AGTR1
SCHEMBL7009867 0.65 AGTR1 (0.50) AGTR1
SCHEMBL6609615 0.65 NPC1 (0.47) SMN1; SMN2TP53HPGDMAPTMEN1
SCHEMBL7016027 0.63 AGTR1 (0.42) AGTR1
SCHEMBL7014690 0.63 AGTR1 (0.42) AGTR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5883111-A STRONG AND LONG-LASTING ACTION BY ORAL ADMINISTRATION; HYPOTENSIVE AGENTS; CARDIOTONIC AGENTS; ALZHEIMER'S DISEASE; TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1999-03-16 US disclosed