SCHEMBL8365166

SCHEMBL8365166

CN(C(=O)[C@@H](N)Cc1ccc(O)cc1)[C@@H](CCCN)C(=O)Nc1ccc2ccccc2c1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MC4R P32245 2/20 0.43
MC5R P33032 2/20 0.43
MC3R P41968 2/20 0.43
F2 P00734 2/20 0.42
OPRD1 P41143 1/20 0.41
BACE1 P56817 2/20 0.39
LTA4H P09960 1/20 0.39
TRPC3 Q13507 1/20 0.39
TRPC7 Q9HCX4 1/20 0.39
TRPC5 Q9UL62 1/20 0.39
KDM4E B2RXH2 2/20 0.38
MEN1 O00255 2/20 0.38
KMT2A Q03164 2/20 0.38
ALDH1A1 P00352 1/20 0.38
CYP1A2 P05177 1/20 0.38
CYP2C19 P33261 1/20 0.38
HIF1A Q16665 1/20 0.38
CHRNA1 P02708 2/20 0.38
CHRNG P07510 2/20 0.38
CHRNB1 P11230 2/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7850361 1.00 MC4R (0.43) MC4RMC5RMC3RF2OPRD1
SCHEMBL7860791 0.93 MC4R (0.48) MC4RMC5RMC3RF2LTA4H
SCHEMBL7857110 0.86 LTA4H (0.45) MC4RMC5RMC3RF2LTA4H
SCHEMBL7857976 0.85 LARS1 (0.46) F2KDM4EMEN1KMT2AALDH1A1
Trifluoroacetic Acid SCHEMBL7857842 0.82 LARS1 (0.42) F2LTA4HCYP1A2MAPTSMN1; SMN2
SCHEMBL8362644 0.81 EPHX1 (0.39) MC4RMC5RMC3RF2KDM4E
SCHEMBL7859247 0.81 EPHX1 (0.39) MC4RMC5RMC3RF2KDM4E
SCHEMBL4610411 0.80 BACE1 (0.57) OPRD1BACE1KDM4EMEN1KMT2A
SCHEMBL29641523 0.78 SLC7A5 (0.52) MC4RMC5RMC3RLNPEP
SCHEMBL29909939 0.78 SLC7A5 (0.52) MC4RMC5RMC3RLNPEP

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1999037667-A1 EFFLUX PUMP INHIBITORS MICROCIDE PHARMACEUTICALS, INC. (US) 1999-07-29 WO disclosed