SCHEMBL8367107

SCHEMBL8367107

CCN1CCOc2cc3c(cc2C1=O)OC1CCCN1C3=O

nearest known ligand 0.70

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
GRIA1 P42261 1/20 0.70
SMN1; SMN2 Q16637 1/20 0.34
PRMT5 O14744 8/20 0.33
WDR77 Q9BQA1 8/20 0.33
NR3C1 P04150 1/20 0.33
PGR P06401 1/20 0.33
AR P10275 1/20 0.33
ROCK2 O75116 3/20 0.32
ROCK1 Q13464 2/20 0.32
GRM5 P41594 1/20 0.32
TNIK Q9UKE5 1/20 0.32
PTGER3 P43115 1/20 0.31
ALPL P05186 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8367566 0.89 GRIA1 (0.64) GRIA1SMN1; SMN2
SCHEMBL678000 0.83 GRIA1 (1.00) GRIA1SMN1; SMN2
SCHEMBL29542563 0.83 GRIA1 (1.00) GRIA1SMN1; SMN2
SCHEMBL8314975 0.83 GRIA1 (0.82) GRIA1
SCHEMBL8368416 0.82 GRIA1 (0.62) GRIA1GRM5
SCHEMBL8368414 0.79 GRIA1 (0.64) GRIA1
SCHEMBL8367555 0.78 GRIA1 (0.80) GRIA1
SCHEMBL8367567 0.78 GRIA1 (0.75) GRIA1
SCHEMBL31562972 0.78 GRIA1 (0.84) GRIA1
SCHEMBL12049626 0.78 GRIA1 (0.84) GRIA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7799913-B2 Carbonylbenzoxazine compounds for enhancing glutamatergic synaptic responses CORTEX PHARMACEUTICALS, INC. (US) 2010-09-21 US disclosed
US-7799913-B2 Carbonylbenzoxazine compounds for enhancing glutamatergic synaptic responses CORTEX PHARMACEUTICALS, INC. (US) 2010-09-21 US disclosed
WO-2003045315-A2 CARBONYLBENZOXAZINE COMPOUNDS FOR ENHANCING GLUTAMATERGIC SYNAPTIC RESPONSES CORTEX PHARMACEUTICALS, INC. (US) 2003-06-05 WO disclosed