SCHEMBL8367127

SCHEMBL8367127

Cc1nnc(C2(c3ccccc3)CCN(C(=O)OCc3ccccc3)CC2)o1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
OPRD1 P41143 9/20 0.56
OPRK1 P41145 5/20 0.56
OPRM1 P35372 1/20 0.51
ALDH1A1 P00352 5/20 0.50
SMN1; SMN2 Q16637 4/20 0.50
ALOX15 P16050 2/20 0.50
GAA P10253 1/20 0.50
MEN1 O00255 3/20 0.49
KMT2A Q03164 3/20 0.49
NPSR1 Q6W5P4 2/20 0.49
L3MBTL1 Q9Y468 1/20 0.47
KDM4E B2RXH2 1/20 0.47
MAPT P10636 1/20 0.47
CYP2C19 P33261 1/20 0.46
HDAC3 O15379 1/20 0.46
HDAC1 Q13547 1/20 0.46
HDAC2 Q92769 1/20 0.46
HDAC6 Q9UBN7 1/20 0.46
NPY1R P25929 1/20 0.46
HSD17B10 Q99714 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4630020 0.88 OPRD1 (0.57) OPRD1OPRK1OPRM1ALDH1A1SMN1; SMN2
SCHEMBL56293 0.75 OPRD1 (0.58) OPRD1OPRK1OPRM1ALDH1A1SMN1; SMN2
SCHEMBL13690026 0.75 MEN1 (0.58) OPRD1OPRK1OPRM1ALDH1A1SMN1; SMN2
SCHEMBL3099492 0.75 OPRD1 (0.48) OPRD1OPRK1OPRM1ALDH1A1SMN1; SMN2
SCHEMBL21581202 0.75 OPRD1 (0.63) OPRD1OPRK1OPRM1MAPT
SCHEMBL2899076 0.75 SMN1; SMN2 (0.57) SMN1; SMN2GAAMEN1KMT2ANPSR1
Hydrochloric Acid SCHEMBL18742622 0.74 OPRD1 (0.57) OPRD1OPRK1OPRM1ALDH1A1SMN1; SMN2
SCHEMBL7556949 0.74 CHRM4 (0.61) OPRD1OPRK1SMN1; SMN2MEN1KMT2A
SCHEMBL1709936 0.74 MEN1 (0.59) OPRD1OPRK1ALDH1A1SMN1; SMN2ALOX15
SCHEMBL541133 0.74 MEN1 (0.63) OPRD1OPRK1ALDH1A1SMN1; SMN2ALOX15

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5965580-A TREATMENT OF SUBSTANCE P- AND NEUROKININ-DEPENDENT DISORDERS SANOFI (FR) 1999-10-12 US disclosed
US-5939411-A PIPERIDINE DERIVATIVES SUBSTITUTED AT POSITION 4 WITH NEW FUNCTIONS OTHER THAN THOSE DESCRIBED PREVIOUSLY HAVE A HIGH AFFINITY FOR NEUROKININ RECEPTORS AND ARE USEFUL FOR TREATMENT OF SUBSTANCE P AND NEUROKININ DEPENDENT PATHOLOGIES SANOFI (FR) 1999-08-17 US disclosed
US-5830906-A Piperidine derivatives, process for obtaining them and pharmaceutical compositions containing them SANOFI (FR) 1998-11-03 US disclosed