SCHEMBL8375808

SCHEMBL8375808

O=C(O)CCCCCCCCCCCCCCC(=O)ON1C(=O)C2C3C=CC(C3)C2C1=O

nearest known ligand 0.55

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
MAPK1 P28482 1/20 0.55
SMN1; SMN2 Q16637 4/20 0.50
L3MBTL1 Q9Y468 1/20 0.50
RAB9A P51151 2/20 0.45
MEN1 O00255 1/20 0.45
KMT2A Q03164 1/20 0.45
ALDH1A1 P00352 5/20 0.43
TDP1 Q9NUW8 1/20 0.42
TSHR P16473 3/20 0.42
USP2 O75604 1/20 0.42
HTT P42858 1/20 0.42
HSD17B10 Q99714 1/20 0.42
PKM P14618 1/20 0.41
HPGD P15428 1/20 0.41
GAA P10253 1/20 0.39
CYP1A2 P05177 1/20 0.39
CYP3A4 P08684 1/20 0.39
CYP2C19 P33261 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4278263 0.94 RAB9A (0.50) MAPK1SMN1; SMN2L3MBTL1RAB9AMEN1
SCHEMBL11752804 0.93 MAPK1 (0.50) MAPK1SMN1; SMN2L3MBTL1RAB9AMEN1
SCHEMBL23476146 0.90 MAPK1 (0.59) MAPK1SMN1; SMN2L3MBTL1RAB9AMEN1
SCHEMBL11296446 0.89 RAB9A (0.45) MAPK1SMN1; SMN2L3MBTL1RAB9AMEN1
SCHEMBL15456601 0.87 MAPK1 (0.46) MAPK1SMN1; SMN2L3MBTL1RAB9AMEN1
SCHEMBL11304940 0.87 MAPK1 (0.48) MAPK1SMN1; SMN2L3MBTL1RAB9AMEN1
SCHEMBL4274070 0.87 MAPK1 (0.53) MAPK1SMN1; SMN2L3MBTL1RAB9AMEN1
SCHEMBL13700584 0.83 SMN1; SMN2 (0.45) MAPK1SMN1; SMN2L3MBTL1RAB9AMEN1
SCHEMBL13599620 0.81 MAPK1 (0.48) MAPK1SMN1; SMN2L3MBTL1RAB9AMEN1
SCHEMBL11298898 0.81 MAPK1 (0.48) MAPK1SMN1; SMN2L3MBTL1RAB9AMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-RE36359-E SUCH AS N-(15-CARBOXYPENTADECANOYLOXY)SUCCINIMIDE; USED TO MODIFY PROTEINS TO OBTAIN PROTEIN DERIVATIVES HAVING IMPROVED BIOAVAILABILITY, NO ANTIGENICITY AND CAN BE ADMINISTERED TO ANIMALS KURARAY CO., LTD. (JP) 1999-10-26 US claimed
US-5414089-A Useful for modifying enzymes or proteins KURARAY CO., LTD. (JP) 1995-05-09 US claimed
US-RE36359-E SUCH AS N-(15-CARBOXYPENTADECANOYLOXY)SUCCINIMIDE; USED TO MODIFY PROTEINS TO OBTAIN PROTEIN DERIVATIVES HAVING IMPROVED BIOAVAILABILITY, NO ANTIGENICITY AND CAN BE ADMINISTERED TO ANIMALS KURARAY CO., LTD. (JP) 1999-10-26 US disclosed
EP-0511600-B1 Long chain carboxylic acid imide ester KURARAY CO (JP) 1999-03-17 EP disclosed
US-5414089-A Useful for modifying enzymes or proteins KURARAY CO., LTD. (JP) 1995-05-09 US disclosed
US-5336782-A N-(carboxyalkoyloxy)succinimides; modifiers of proteins and enzymes to prolong their plasma half-lives; nontoxic; antitumor and -carcinogenic agents KURARAY CO., LTD. (JP) 1994-08-09 US disclosed
EP-0511600-A2 Long chain carboxylic acid imide ester KURARAY CO., LTD. (JP) 1992-11-04 EP disclosed