SCHEMBL8375869

SCHEMBL8375869

CN(C)c1cccc(Oc2ncc(F)c(N(C)C(Oc3cccc(C#N)c3)C(=O)O)c2F)c1

nearest known ligand 0.39

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
PTGER4 P35408 1/20 0.39
PTGER2 P43116 1/20 0.39
F10 P00742 5/20 0.38
F2 P00734 3/20 0.38
DCK P27707 1/20 0.37
HRH3 Q9Y5N1 1/20 0.37
F3 P13726 2/20 0.36
PLG P00747 2/20 0.36
PLAU P00749 2/20 0.36
F7 P08709 1/20 0.35
HAO1 Q9UJM8 3/20 0.35
JAK2 O60674 1/20 0.35
JAK1 P23458 1/20 0.35
JAK3 P52333 1/20 0.35
GCK P35557 1/20 0.34
NOD1 Q9Y239 1/20 0.34
APP P05067 1/20 0.34
PLAT P00750 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8333175 0.79 F10 (0.46) F10F2F3
SCHEMBL6579150 0.76 F10 (0.51) F10F2F3PLGPLAU
SCHEMBL6579247 0.71 F10 (0.65) F10F2F3F7
SCHEMBL6578477 0.67 F10 (0.51) F10F2PLGPLAUHAO1
SCHEMBL6581900 0.65 F10 (0.55) F10F2F3F7
SCHEMBL7074510 0.64 APP (0.41) F10F2GCKAPP
SCHEMBL6576219 0.64 F10 (0.60) F10F2F3PLGPLAU
SCHEMBL6578924 0.64 F10 (0.66) F10F2F3PLGPLAU
SCHEMBL6579054 0.63 F10 (0.70) F10F2F3F7
SCHEMBL6576475 0.62 F10 (0.72) F10F2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5889005-A Benzamidine derivatives and their use for treating thrombotic diseases BERLEX LABORATORIES, INC. (US) 1999-03-30 US disclosed
US-5883100-A Benzamidine derivatives and their use as anti-coagulants BERLEX LABORATORIES, INC. (US) 1999-03-16 US disclosed
US-5877181-A Benzamidine derivatives and their use as anti-coagulants BERLEX LABORATORIES, INC. (US) 1999-03-02 US disclosed
US-5691364-A Benzamidine derivatives and their use as anti-coagulants BERLEX LABORATORIES, INC. (US) 1997-11-25 US disclosed