SCHEMBL8376192

SCHEMBL8376192

CN1C(=O)C=C[C@@]2(C)C1CC[C@@H]1[C@H]2CC[C@]2(C)C(C(=O)NC(C)(c3ccccc3)C(F)(F)F)CC[C@@H]12

nearest known ligand 0.74

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
SRD5A2 P31213 4/20 0.71
SRD5A1 P18405 3/20 0.71
AR P10275 4/20 0.69
KCNH2 Q12809 2/20 0.51
LMNA P02545 2/20 0.49
CYP3A4 P08684 2/20 0.49
CYP2C9 P11712 2/20 0.49
CYP2C19 P33261 2/20 0.49
ABCC4 O15439 1/20 0.49
ABCB11 O95342 1/20 0.49
ADORA3 P0DMS8 1/20 0.49
CHRM1 P11229 1/20 0.49
HSD3B1 P14060 1/20 0.49
NFKB1 P19838 1/20 0.49
MAPK1 P28482 1/20 0.49
THPO P40225 1/20 0.49
BLM P54132 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8376189 1.00 SRD5A2 (0.71) SRD5A2SRD5A1ARKCNH2LMNA
SCHEMBL8074134 0.91 SRD5A2 (0.70) SRD5A2SRD5A1ARKCNH2
SCHEMBL8074137 0.91 SRD5A2 (0.70) SRD5A2SRD5A1ARKCNH2
SCHEMBL9022541 0.90 AR (0.68) SRD5A2SRD5A1ARKCNH2LMNA
SCHEMBL9022270 0.90 AR (0.68) SRD5A2SRD5A1ARKCNH2LMNA
SCHEMBL9022263 0.90 AR (0.68) SRD5A2SRD5A1ARKCNH2LMNA
SCHEMBL9022545 0.90 AR (0.68) SRD5A2SRD5A1ARKCNH2LMNA
SCHEMBL5212103 0.89 AR (0.67) SRD5A2SRD5A1ARKCNH2LMNA
SCHEMBL10521077 0.85 AR (0.67) SRD5A2SRD5A1ARKCNH2LMNA
SCHEMBL7790540 0.85 AR (0.67) SRD5A2SRD5A1ARKCNH2LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0902790-A1 PROCESS FOR PREPARING STEROIDS HAVING A CARBOXAMIDE SIDE-CHAIN PHARMACIA & UPJOHN S.p.A. (IT) 1999-03-24 EP disclosed
WO-1997040062-A1 PROCESS FOR PREPARING STEROIDS HAVING A CARBOXAMIDE SIDE-CHAIN PHARMACIA & UPJOHN S.P.A. (IT) 1997-10-30 WO disclosed