SCHEMBL8388609

SCHEMBL8388609

Cc1csc(C2=C(c3ccc(S(C)(=O)=O)nc3)CC3(CCC3)C2)c1

nearest known ligand 0.44

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 17/20 0.44
PTGS1 P23219 8/20 0.41
PIK3CD O00329 1/20 0.36
PIP5K1C O60331 1/20 0.36
PIK3CB P42338 1/20 0.36
PI4KA P42356 1/20 0.36
PIK3CG P48736 1/20 0.36
PI4KB Q9UBF8 1/20 0.36
ALOX5AP P20292 1/20 0.36
GRIN2B Q13224 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8383973 0.98 PTGS2 (0.44) PTGS2PTGS1PIK3CDPIP5K1CPIK3CB
SCHEMBL8385117 0.95 PTGS2 (0.46) PTGS2PTGS1PIK3CDPIP5K1CPIK3CB
SCHEMBL8388351 0.88 PTGS2 (0.41) PTGS2PTGS1GRIN2B
SCHEMBL8389075 0.85 PTGS2 (0.41) PTGS2PTGS1
SCHEMBL8383787 0.85 PTGS2 (0.58) PTGS2PTGS1ALOX5AP
SCHEMBL8388744 0.84 PTGS2 (0.64) PTGS2PTGS1
SCHEMBL8386204 0.82 PTGS2 (0.58) PTGS2PTGS1ALOX5AP
SCHEMBL8386008 0.81 PTGS2 (0.64) PTGS2PTGS1
SCHEMBL8384244 0.81 PTGS2 (0.67) PTGS2PTGS1
SCHEMBL8384032 0.80 PTGS2 (0.51) PTGS2PTGS1ALOX5AP

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0743938-B1 SUBSTITUTED SPIRO COMPOUNDS FOR THE TREATMENT OF INFLAMMATION SEARLE & CO (US) 1999-04-21 EP disclosed
US-5393790-A Diphenyl- or phenyl/pyridyl-substituted spiroheptenes, -octenes,-nonenes or -decenes; cyclooxygenase II inhibitors; side effect reduction; antipyretics; antiarthritic agents G.D. SEARLE & CO. (US) 1995-02-28 US disclosed