SCHEMBL8397140

SCHEMBL8397140

COc1ccc(Cl)c(Oc2c(NS(=O)(=O)c3ccc(C(C)(C)C)cc3)nc(C)nc2OCCOC(C)=O)c1

nearest known ligand 0.62

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
EDNRA P25101 16/20 0.62
EDNRB P24530 14/20 0.62
ABCC3 O15438 1/20 0.49
ABCC4 O15439 1/20 0.49
NR1I2 O75469 1/20 0.49
ABCB11 O95342 1/20 0.49
DHPS P49366 1/20 0.49
NR1H3 Q13133 1/20 0.49
NR1I3 Q14994 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8399577 0.91 EDNRA (0.61) EDNRAEDNRBABCC3ABCC4NR1I2
SCHEMBL7305595 0.91 EDNRA (0.74) EDNRAEDNRBABCC3ABCC4NR1I2
SCHEMBL8397146 0.90 EDNRA (0.60) EDNRAEDNRBABCC3ABCC4NR1I2
SCHEMBL7597077 0.90 EDNRA (0.60) EDNRAEDNRB
SCHEMBL7295822 0.88 EDNRA (0.78) EDNRAEDNRBABCC3ABCC4NR1I2
SCHEMBL9156436 0.87 EDNRA (0.59) EDNRAEDNRB
SCHEMBL8327410 0.83 EDNRA (0.57) EDNRAEDNRBABCC3ABCC4NR1I2
SCHEMBL7017153 0.83 EDNRA (0.57) EDNRAEDNRB
SCHEMBL7293947 0.83 EDNRA (0.56) EDNRAEDNRB
SCHEMBL795564 0.82 EDNRA (0.71) EDNRAEDNRBABCC3ABCC4NR1I2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5856484-A Sulfonylaminopyrimidine carboxylic acid derivatives having endothelin inhibiting activity HOFFMANN-LA ROCHE INC. (US) 1999-01-05 US disclosed