SCHEMBL8397155

SCHEMBL8397155

O=C(O)C(c1ccc(F)cc1F)c1ccc(F)cc1F

nearest known ligand 0.67

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CES2 O00748 4/20 0.53
CES1 P23141 4/20 0.53
IDO1 P14902 1/20 0.42
TDO2 P48775 1/20 0.42
ALDH1A1 P00352 3/20 0.39
HTT P42858 2/20 0.39
CYP2C19 P33261 1/20 0.39
NPC1 O15118 1/20 0.39
RAB9A P51151 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.39
KEAP1 Q14145 1/20 0.38
KCNN4 O15554 1/20 0.38
KDM4E B2RXH2 1/20 0.38
MEN1 O00255 1/20 0.38
USP2 O75604 1/20 0.38
DHFR P00374 1/20 0.38
CA1 P00915 1/20 0.38
CA2 P00918 1/20 0.38
LMNA P02545 1/20 0.38
TTR P02766 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3703093 0.83 CES2 (0.53) CES2CES1IDO1TDO2ALDH1A1
SCHEMBL3065996 0.83 CES2 (0.53) CES2CES1IDO1TDO2ALDH1A1
SCHEMBL19183094 0.82 KDM4E (0.40) CES2CES1IDO1TDO2HTT
SCHEMBL29658750 0.82 CES2 (0.66) CES2CES1IDO1TDO2ALDH1A1
SCHEMBL1671155 0.82 CES2 (0.66) CES2CES1IDO1TDO2ALDH1A1
SCHEMBL1671151 0.82 CES2 (0.66) CES2CES1IDO1TDO2ALDH1A1
SCHEMBL1115280 0.80 CES2 (0.50) CES2CES1IDO1TDO2ALDH1A1
SCHEMBL31117279 0.80 PTGS1 (0.54) CES2CES1CYP2C19MEN1LMNA
SCHEMBL30882180 0.80 CES2 (0.50) CES2CES1IDO1TDO2ALDH1A1
SCHEMBL19182930 0.80 PTGS1 (0.54) CES2CES1CYP2C19MEN1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5955501-A DERIVED FROM PHORBOIDS OF THE DITERPENE- AND BENZOLACTAM-CLASSES. PROCYON PHARMACEUTICALS, INC. (US) 1999-09-21 US disclosed
US-5891870-A ANTIINFLAMMATORY AGENTS USING BENZODITERPENES AND BENZOLACTAMS PROCYON PHARMACEUTICALS, INC. (US) 1999-04-06 US disclosed
US-5891906-A Polyacetate-derived phorboids having anti-inflammatory and other uses PROCYON PHARMACEUTICALS, INC. (US) 1999-04-06 US disclosed
US-5886019-A REPLACEMENT OF HYDROXYMETHYL OR-ETHYL GROUP ON TRICYCLIC AROMATIC HETEROCYCLIC COMPOUNDS HAVING INDOLE, INDENE, BENZOFURAN OR BENZOTHIOPHENE SKELETON; ANTIINFLAMMATORY, ANTIVIRAL PROCYON PHARMACEUTICALS, INC. (US) 1999-03-23 US disclosed
US-5750568-A DITERPENE PHORBOIDS PROCYON PHARMACEUTICALS, INC. (US) 1998-05-12 US disclosed
US-5716968-A ANTIINFLAMMATORY AGENTS; VIRICIDE PROCYON PHARMACEUTICALS, INC. (US) 1998-02-10 US disclosed