SCHEMBL8398115

SCHEMBL8398115

CC(C)(C)OC(=O)N[C@H]1CCC[C@H]1Cc1ccc(OCc2ccccc2)cc1

nearest known ligand 0.47

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 4/20 0.47
L3MBTL1 Q9Y468 1/20 0.47
CYSLTR2 Q9NS75 1/20 0.46
CYSLTR1 Q9Y271 1/20 0.46
YAP1 P46937 3/20 0.44
RAB9A P51151 2/20 0.43
SMN1; SMN2 Q16637 2/20 0.43
NPC1 O15118 1/20 0.43
MEN1 O00255 2/20 0.42
KDM4C Q9H3R0 1/20 0.42
BCL2 P10415 1/20 0.42
HTR2C P28335 1/20 0.42
HTR2B P41595 1/20 0.42
MME P08473 1/20 0.42
HDAC1 Q13547 1/20 0.42
KDM4E B2RXH2 2/20 0.42
LTA4H P09960 1/20 0.42
MAPT P10636 1/20 0.42
PPARA Q07869 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7377064 1.00 KMT2A (0.47) KMT2AL3MBTL1CYSLTR2CYSLTR1YAP1
SCHEMBL8398113 1.00 KMT2A (0.47) KMT2AL3MBTL1CYSLTR2CYSLTR1YAP1
SCHEMBL7328301 0.82 NPC1 (0.41) KMT2AL3MBTL1YAP1RAB9ASMN1; SMN2
SCHEMBL8654091 0.82 NPC1 (0.41) KMT2AL3MBTL1YAP1RAB9ASMN1; SMN2
SCHEMBL8650717 0.82 NPC1 (0.41) KMT2AL3MBTL1YAP1RAB9ASMN1; SMN2
SCHEMBL7337139 0.82 NPC1 (0.41) KMT2AL3MBTL1YAP1RAB9ASMN1; SMN2
SCHEMBL7375317 0.80 HRH3 (0.48) KMT2ACYSLTR2CYSLTR1RAB9ANPC1
SCHEMBL7375323 0.80 HRH3 (0.48) KMT2ACYSLTR2CYSLTR1RAB9ANPC1
SCHEMBL7375321 0.80 HRH3 (0.48) KMT2ACYSLTR2CYSLTR1RAB9ANPC1
Hydrochloric Acid SCHEMBL8395630 0.79 HRH3 (0.47) KMT2ACYSLTR2CYSLTR1RAB9ANPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0752981-B1 SUBSTITUTED CYCLOPENTYLAMINE DERIVATIVES AND THEIR USE AS CALCIUM CHANNEL ANTAGONISTS SMITHKLINE BEECHAM PLC (GB) 1999-06-09 EP disclosed
US-5817698-A Substituted cycloalkylamine derivatives and their use as calcium channel antagonists SMITHKLINE BEECHAM PLC (GB) 1998-10-06 US disclosed