SCHEMBL8398557

SCHEMBL8398557

Cc1ccc(O)c(C)c1NC(=O)C[C@H]1CCCN1

nearest known ligand 0.42

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
ADORA2A P29274 1/20 0.42
FLT3 P36888 1/20 0.40
KHK P50053 1/20 0.37
CHRNB4 P30926 2/20 0.35
CHRNA3 P32297 2/20 0.35
HSP90AA1 P07900 1/20 0.35
HSP90AB1 P08238 1/20 0.35
KDM4E B2RXH2 1/20 0.34
HTT P42858 1/20 0.34
GHSR Q92847 1/20 0.34
IL1B P01584 1/20 0.34
MEN1 O00255 1/20 0.33
RAB9A P51151 1/20 0.33
KMT2A Q03164 1/20 0.33
PBK Q96KB5 1/20 0.33
FPR3 P25089 1/20 0.33
FPR2 P25090 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8397261 1.00 ADORA2A (0.42) ADORA2AFLT3KHKCHRNB4CHRNA3
SCHEMBL8393468 1.00 ADORA2A (0.42) ADORA2AFLT3KHKCHRNB4CHRNA3
SCHEMBL2096759 0.81 EPHX1 (0.48) ADORA2AKHKMEN1KMT2A
SCHEMBL11036183 0.80 EPHX1 (0.50) KHKMEN1KMT2A
SCHEMBL6242633 0.71 SCN1A (0.33) HTTMEN1KMT2A
SCHEMBL7124281 0.70 TERT (0.42) KDM4EHTTMEN1KMT2A
SCHEMBL8398430 0.69 CA1 (0.43) KDM4EHTTMEN1KMT2A
SCHEMBL719291 0.68 ADORA2A (0.40) ADORA2AFLT3KHKHTTGHSR
SCHEMBL714038 0.68 ADORA2A (0.40) ADORA2AFLT3KHKHTTGHSR
SCHEMBL7259516 0.68 EPHX2 (0.61) ADORA2AKHKRAB9AKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0915834-A1 METHOD AND COMPOSITIONS FOR PRODUCING ANALGESIA ELAN PHARMACEUTICALS, INC. (US) 1999-05-19 EP claimed
WO-1997033860-A1 METHOD AND COMPOSITIONS FOR PRODUCING ANALGESIA NEUREX CORPORATION (US) 1997-09-18 WO claimed
EP-0915834-A1 METHOD AND COMPOSITIONS FOR PRODUCING ANALGESIA ELAN PHARMACEUTICALS, INC. (US) 1999-05-19 EP disclosed
WO-1997033860-A1 METHOD AND COMPOSITIONS FOR PRODUCING ANALGESIA NEUREX CORPORATION (US) 1997-09-18 WO disclosed