SCHEMBL8401002

SCHEMBL8401002

O=C(O)c1ccccc1OCCN1CCCCC1

nearest known ligand 0.75

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
DRD2 P14416 2/20 0.75
DRD1 P21728 2/20 0.75
DRD3 P35462 2/20 0.75
KMT2A Q03164 2/20 0.72
MEN1 O00255 1/20 0.72
GAA P10253 1/20 0.72
ABCB1 P08183 7/20 0.70
MAPT P10636 1/20 0.66
KDM4E B2RXH2 2/20 0.65
SMN1; SMN2 Q16637 1/20 0.65
TSHR P16473 1/20 0.60
HRH1 P35367 2/20 0.58
DRD4 P21917 1/20 0.58
DRD5 P21918 1/20 0.58
ALDH1A1 P00352 2/20 0.58
PTK2B Q14289 1/20 0.58
TDP1 Q9NUW8 1/20 0.57

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11365759 1.00 DRD2 (0.75) DRD2DRD1DRD3KMT2AMEN1
Hydrochloric Acid SCHEMBL8665681 0.99 DRD2 (0.73) DRD2DRD1DRD3KMT2AMEN1
SCHEMBL11336084 0.93 MAPT (0.76) DRD2DRD1DRD3KMT2AMEN1
SCHEMBL11712364 0.90 DRD2 (0.72) DRD2DRD1DRD3KMT2AMEN1
SCHEMBL11801298 0.90 DRD2 (0.72) DRD2DRD1DRD3KMT2AMEN1
SCHEMBL11712503 0.90 DRD2 (0.72) DRD2DRD1DRD3KMT2AMEN1
SCHEMBL11730898 0.90 DRD2 (0.72) DRD2DRD1DRD3KMT2AMEN1
SCHEMBL11804646 0.88 DRD2 (0.74) DRD2DRD1DRD3KMT2AMEN1
SCHEMBL8639351 0.87 KDM4E (0.68) DRD2DRD1DRD3KMT2AMEN1
SCHEMBL876068 0.87 DRD2 (0.69) DRD2DRD1DRD3KMT2AMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5955608-A Process for preparing benzoic acid derivative intermediates and benzothiophene pharmaceutical agents ELI LILLY AND COMPANY (US) 1999-09-21 US disclosed
EP-0699673-B1 Process for preparing benzoic acid derivative intermediates and benzothiophene pharmaceutical agents LILLY CO ELI (US) 1998-04-22 EP disclosed
US-5731436-A Process for preparing benzoic acid derivative intermediates and benzothiophene pharmaceutical agents ELI LILLY AND COMPANY (US) 1998-03-24 US disclosed
EP-0699673-A1 Process for preparing benzoic acid derivative intermediates and benzothiophene pharmaceutical agents ELI LILLY AND COMPANY (US) 1996-03-06 EP disclosed
US-4298603-A LOCAL ANESTHETICS INDUSTRIAL TECHNOLOGY RESEARCH INSTITUTE (TW) 1981-11-03 US disclosed
EP-0031632-A1 O-Aminoalkylsalicylates, process for their preparation, and their pharmaceutical compositions INDUSTRIAL TECHNOLOGY RESEARCH INSTITUTE (TW) 1981-07-08 EP disclosed