Benzene

Benzene

SCHEMBL8401598

CCc1cn(CC(=O)O)c(=O)c(C(=O)CCc2ccccc2)c1N.c1ccccc1

nearest known ligand 0.40

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Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
GAA P10253 1/20 0.40
MAPT P10636 1/20 0.40
SLC5A1 P13866 1/20 0.40
SLC5A2 P31639 1/20 0.40
ALDH1A1 P00352 2/20 0.39
RXFP1 Q9HBX9 1/20 0.39
ABCB1 P08183 9/20 0.39
KEAP1 Q14145 1/20 0.39
ADORA2A P29274 1/20 0.38
FFAR1 O14842 1/20 0.37
PLA2G4A P47712 1/20 0.37
NPC1 O15118 1/20 0.36
RAB9A P51151 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27465499 0.71 KMT2A (0.40) GAAMAPTALDH1A1ADORA2ANPC1
Benzene SCHEMBL8401599 0.67 TSHR (0.48) GAAMAPTALDH1A1NPC1RAB9A
SCHEMBL7483874 0.66 HDAC1 (0.41) MAPTALDH1A1RXFP1KEAP1
SCHEMBL19873809 0.65 PDE3B (0.46) MAPTALDH1A1RXFP1
SCHEMBL12303227 0.64 ABCB1 (0.54) GAAMAPTSLC5A1SLC5A2ALDH1A1
SCHEMBL4989754 0.63 KDM4E (0.49) MAPTALDH1A1
Phenyl Propionic Acid SCHEMBL29473504 0.62 KEAP1 (0.95) MAPTALDH1A1RXFP1KEAP1FFAR1
Phenyl Propionic Acid SCHEMBL6534964 0.62 KEAP1 (0.95) MAPTALDH1A1RXFP1KEAP1FFAR1
Phenyl Propionic Acid SCHEMBL14715905 0.62 KEAP1 (0.95) MAPTALDH1A1RXFP1KEAP1FFAR1
SCHEMBL12874520 0.62 KMT2A (0.66) GAAMAPTALDH1A1RXFP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5973111-A NOVEL COMPOUNDS THAT ARE CAPABLE OF BINDING TO THE ACTIVE SITE OF INTERLEUKIN-1B-CONVERTING ENZYME (ICE) AND INHIBITING ACTIVITY OF THAT ENZYME; ADMINISTERING TO TREAT INFLAMMATORY, AUTOIMMUNE, AND NEURODEGENERATIVE DISEASES VERTEX PHARMACEUTICALS, INC. (US) 1999-10-26 US disclosed